日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

TSPO Modulation Prevents Photoreceptor Degeneration and Produces Neuroprotective Effects in an Animal Model of Retinitis Pigmentosa

TSPO调节可预防视网膜色素变性动物模型中的光感受器退化并产生神经保护作用

Corsi, Francesca; Castagnoli, Jacopo; Galante, Alessia; Fabiano, Angela; Nuti, Elisa; Piras, Anna Maria; Taliani, Sabrina; Piano, Ilaria; Gargini, Claudia

The protease ADAMTS5 controls ovarian cancer cell invasion, downstream of Rab25.

蛋白酶ADAMTS5控制卵巢癌细胞的侵袭,位于Rab25的下游

Yuan Shengnan, Bacchetti Rachele, Adams Jamie, Cuffaro Doretta, Rossello Armando, Nuti Elisa, Santamaria Salvatore, Rainero Elena

Anti-tumor efficacy and Vδ2 T-cell activation via EGFR antibody-drug conjugates featuring novel aminobisphosphonates

新型氨基双膦酸盐类EGFR抗体药物偶联物发挥抗肿瘤功效并激活Vδ2 T细胞

Cuffaro, Doretta; Di Gregorio, Linda; Mangini, Camilla; Taglieri, Martina; Matis, Serena; Benelli, Roberto; Ardy, Massimo; Salvini, Laura; Rossello, Armando; Poggi, Alessandro; Raffaghello, Lizzia; Nuti, Elisa

Design, synthesis and biological activity of glycoconjugated ADAMTS5 exosite inhibitors: applications in osteoarthritis and ovarian cancer models.

糖缀合ADAMTS5外位点抑制剂的设计、合成和生物活性:在骨关节炎和卵巢癌模型中的应用。

Cuffaro Doretta, Blagg Sophie, Yamamoto Kazuhiro, Pinzi Luca, Bacchetti Rachele, Yuan Shengnan, Tew Simon, Campagnolo Paola, D'Andrea Felicia, Crispino Enrico, Rastelli Giulio, Rossello Armando, Rainero Elena, Nuti Elisa, Santamaria Salvatore

Identification of novel N-benzyloxy-amino acid hydroxamates as inhibitors of the virulence factor LasB from Pseudomonas aeruginosa.

鉴定出新型 N-苄氧基氨基酸羟肟酸酯类化合物可作为铜绿假单胞菌毒力因子 LasB 的抑制剂

Di Leo Riccardo, Crispino Enrico, Cuffaro Doretta, Maisetta Giuseppantonio, Bertacca Andrea, Bianchi Marta, Batoni Giovanna, Wushur Imin, Rahman Fatema Amatur, Winberg Jan-Olof, Sylte Ingebrigt, Rossello Armando, Nuti Elisa

A series of benzensulfonamide derivatives as new potent carbonic anhydrase IX and XII inhibitors

一系列苯磺酰胺衍生物作为新型强效碳酸酐酶IX和XII抑制剂

Nencetti, Susanna; Cuffaro, Doretta; Ciccone, Lidia; Nocentini, Alessio; Di Stefano, Miriana; Poli, Giulio; Macchia, Marco; Tuccinardi, Tiziano; Nuti, Elisa; Supuran, Claudiu T; Rossello, Armando; Orlandini, Elisabetta

New isoxazolidinyl-based N-alkylethanolamines as new activators of human brain carbonic anhydrases

新型异噁唑烷基N-烷基乙醇胺作为人脑碳酸酐酶的新型激活剂

Cuffaro, Doretta; Di Leo, Riccardo; Ciccone, Lidia; Nocentini, Alessio; Supuran, Claudiu T; Nuti, Elisa; Rossello, Armando

Effective bioremediation of clarithromycin and diclofenac in wastewater by microbes and Arundo donax L

微生物和芦竹对废水中的克拉霉素和双氯芬酸进行有效生物修复

Laura Ercoli, Rudy Rossetto, Sabrina Di Giorgi, Andrea Raffaelli, Marco Nuti, Elisa Pellegrino

Inhibitors of ADAM10 reduce Hodgkin lymphoma cell growth in 3D microenvironments and enhance brentuximab-vedotin effect

ADAM10抑制剂可减少3D微环境中霍奇金淋巴瘤细胞的生长,并增强brentuximab-vedotin的疗效。

Pece, Roberta; Tavella, Sara; Costa, Delfina; Varesano, Serena; Camodeca, Caterina; Cuffaro, Doretta; Nuti, Elisa; Rossello, Armando; Alfano, Massimo; D'Arrigo, Cristina; Galante, Denise; Ravetti, Jean-Louis; Gobbi, Marco; Tosetti, Francesca; Poggi, Alessandro; Zocchi, Maria Raffaella

Targeting Aggrecanases for Osteoarthritis Therapy: From Zinc Chelation to Exosite Inhibition

靶向聚集蛋白酶治疗骨关节炎:从锌螯合到外位点抑制

Cuffaro, Doretta; Ciccone, Lidia; Rossello, Armando; Nuti, Elisa; Santamaria, Salvatore