日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of potent BET bromodomain 1 stereoselective inhibitors using DNA-encoded chemical library selections

利用DNA编码化学库筛选发现强效BET溴结构域1立体选择性抑制剂

Modukuri, Ram K; Yu, Zhifeng; Tan, Zhi; Ta, Hai Minh; Ucisik, Melek Nihan; Jin, Zhuang; Anglin, Justin L; Sharma, Kiran L; Nyshadham, Pranavanand; Li, Feng; Riehle, Kevin; Faver, John C; Duong, Kevin; Nagarajan, Sureshbabu; Simmons, Nicholas; Palmer, Stephen S; Teng, Mingxing; Young, Damian W; Yi, Joanna S; Kim, Choel; Matzuk, Martin M

Discovery and characterization of bromodomain 2-specific inhibitors of BRDT

BRDT溴结构域2特异性抑制剂的发现与表征

Yu, Zhifeng; Ku, Angela F; Anglin, Justin L; Sharma, Rajesh; Ucisik, Melek Nihan; Faver, John C; Li, Feng; Nyshadham, Pranavanand; Simmons, Nicholas; Sharma, Kiran L; Nagarajan, Sureshbabu; Riehle, Kevin; Kaur, Gundeep; Sankaran, Banumathi; Storl-Desmond, Marta; Palmer, Stephen S; Young, Damian W; Kim, Choel; Matzuk, Martin M

DNA-encoded chemistry technology yields expedient access to SARS-CoV-2 M(pro) inhibitors.

DNA编码化学技术可快速获得SARS-CoV-2 M(pro)抑制剂

Chamakuri Srinivas, Lu Shuo, Ucisik Melek Nihan, Bohren Kurt M, Chen Ying-Chu, Du Huang-Chi, Faver John C, Jimmidi Ravikumar, Li Feng, Li Jian-Yuan, Nyshadham Pranavanand, Palmer Stephen S, Pollet Jeroen, Qin Xuan, Ronca Shannon E, Sankaran Banumathi, Sharma Kiran L, Tan Zhi, Versteeg Leroy, Yu Zhifeng, Matzuk Martin M, Palzkill Timothy, Young Damian W

Discovery of potent thrombin inhibitors from a protease-focused DNA-encoded chemical library

从以蛋白酶为靶点的DNA编码化合物库中发现强效凝血酶抑制剂

Dawadi, Surendra; Simmons, Nicholas; Miklossy, Gabriella; Bohren, Kurt M; Faver, John C; Ucisik, Melek Nihan; Nyshadham, Pranavanand; Yu, Zhifeng; Matzuk, Martin M

Identifying Oxacillinase-48 Carbapenemase Inhibitors Using DNA-Encoded Chemical Libraries

利用DNA编码化合物库鉴定奥沙西林酶-48碳青霉烯酶抑制剂

Taylor, Doris Mia; Anglin, Justin; Park, Suhyeorn; Ucisik, Melek N; Faver, John C; Simmons, Nicholas; Jin, Zhuang; Palaniappan, Murugesan; Nyshadham, Pranavanand; Li, Feng; Campbell, James; Hu, Liya; Sankaran, Banumathi; Prasad, B V Venkataram; Huang, Hongbing; Matzuk, Martin M; Palzkill, Timothy

Homogeneous and Functional Group Tolerant Ring-Closing Metathesis for DNA-Encoded Chemical Libraries

用于DNA编码化学库的均相和官能团耐受的闭环复分解反应

Monty, Olivier B C; Nyshadham, Pranavanand; Bohren, Kurt M; Palaniappan, Murugesan; Matzuk, Martin M; Young, Damian W; Simmons, Nicholas