日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Utilizing the HiBiT System to Identify CARM1 Degraders for Targeted Cancer Therapy

利用HiBiT系统鉴定CARM1降解剂用于靶向癌症治疗

Bacabac, Megan; Hu, Mingshan; Liu, Fabao; Kim, Eui-Jun; Grkovic, Tanja; Kumar, Rohitesh; Akee, Rhone K; Hayes, Isaac; Mudududdla, Ramesh; Wang, Yidan; McGuire, Mason; Tang, Weiping; O'Keefe, Barry R; Bugni, Tim S; Xu, Wei

Exploring the chemodiversity of antimicrobial minalemines from Didemnum granulatum by neutral loss graph

利用中性损失图探索Didemnum granulatum中抗菌minalemines的化学多样性

Freire, Vítor F; Evans, Jason R; Martínez-Fructuoso, Lucero; Kumar, Rohitesh; Akee, Rhone K; Hogan, Svetlana; Thornburg, Christopher C; Peyser, Brian D; Ensel, Susan; Wang, Dongdong; Grkovic, Tanja; O'Keefe, Barry R

Gonystylones A-E, Antiproliferative 5,6-Dihydro-α-pyrones from the Plant Gonystylus borneensis

Gonystylones AE,一种来自植物 Gonystylus borneensis 的抗增殖性 5,6-二氢-α-吡喃酮类化合物。

Kim, Chang-Kwon; Freire, Vitor F; Dey, Soumili; Woldemichael, Girma M; Kim, Yong Yean; Wen, Xinyu; Chou, Hsien-Chao; Song, Young K; Wei, Jun S; Akee, Rhone K; Orfanoudaki, Maria; Dalilian, Masoumeh; Khan, Javed; Grkovic, Tanja; O'Keefe, Barry R

DeepTarget predicts anti-cancer mechanisms of action of small molecules by integrating drug and genetic screens

DeepTarget通过整合药物筛选和基因筛选来预测小分子抗癌作用机制。

Sinha, Sanju; Sinha, Neelam; Perales, Marlenne; Tarrab, Adi; Nguyen, Trinh; Liu, Lihe; Cantore, Thomas; Alvarez, Kyle; Patiyal, Sumeet; Mukherjee, Sumit; Madan, Sanna; Tharp, Kevin; Zhao, Jianhua; Kumar, Ranjit; Flanigan, Greg; Beutler, John A; O'Keefe, Barry R; Meerzaman, Daoud; Ben-David, Uri; Deshpande, Aniruddha J; Ruppin, Eytan

Antiproliferative cassaine diterpenoid amines from the leaves and twigs of the traditional Thai medicinal plant Erythrophleum teysmannii (Kurz) Craib

从泰国传统药用植物 Erythrophleum teysmannii (Kurz) Craib 的叶和枝中提取的抗增殖卡赛因二萜胺类化合物

Orfanoudaki, Maria; Wang, Dongdong; Du, Lin; Ruchirawat, Somsak; Kittakoop, Prasat; Grkovic, Tanja; Mahidol, Chulabhorn; O'Keefe, Barry R

ShiftScan: A tool for rapid analysis of high-throughput differential scanning fluorimetry data and compound prioritization

ShiftScan:一种用于快速分析高通量差示扫描荧光数据和化合物优先级排序的工具

Waterworth, Samantha C; Shenoy, Shilpa R; Sharma, Nirmala D; Wolcott, Chris; Donohue, Duncan E; O'Keefe, Barry R; Beutler, John A

A Biosynthetic and Taxonomic Atlas of the Global Lichen Holobiont

全球地衣全生物体的生物合成和分类图谱

Waterworth, Samantha C; Egbert, Susan; Sorensen, John; O'Keefe, Barry R; Beutler, John A

Biochemical and biophysical characterization of inositol-tetrakisphosphate 1-kinase inhibitors.

肌醇四磷酸1-激酶抑制剂的生化和生物物理特性

Ng Martin Y, Wang Huanchen, Zhang Haibo, Prucker Isabel, Perera Lalith, Goncharova Ekaterina, Wamiru Antony, Jessen Henning J, Stanley Robin E, Shears Stephen B, Luo Ji, O'Keefe Barry R, Wilson Brice A P

Isolation and structure elucidation of Dm-CVNH, a new cyanovirin-N homolog with activity against SARS-CoV-2 and HIV-1.

从 SARS-CoV-2 和 HIV-1 中分离和解析出新型氰基病毒素-N 同系物 Dm-CVNH 的结构

Orfanoudaki Maria, Krumpe Lauren R H, Shenoy Shilpa R, Wilson Jennifer, Guszczynski Tad, Henrich Curtis J, Temme J Sebastian, Gildersleeve Jeffrey C, Molina-Molina Elisa, Erkizia Itziar, Blanco JuliÃ, Izquierdo-Useros Nuria, Montiero Fabio, Tanuri Amilcar, Rech Elibio, O'Keefe Barry R

Identification of Cembrane Diterpenoids from Sinularia sp. That Reduce the Viability of Diffuse Pleural Mesothelioma Cell Lines

从Sinularia sp.中鉴定出能降低弥漫性胸膜间皮瘤细胞系活力的Cembrane二萜类化合物

Orfanoudaki, Maria; Shaikh, Anam F; Wang, Dongdong; Singh, Vivek; Du, Lin; Wilson, Jennifer A; Wamiru, Antony; Goncharova, Ekaterina I; Pruett, Nathanael; Hoang, Chuong D; Wilson, Brice A P; O'Keefe, Barry R