Target Identification with Live-Cell Photoaffinity Labeling and Mechanism of Action Elucidation of ARN23765, a Highly Potent CFTR Corrector.
利用活细胞光亲和标记进行靶标鉴定和高效 CFTR 校正剂 ARN23765 的作用机制阐明
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c02654
Romeo Elisa, Saccoliti Francesco, Ocello Riccardo, Andonaia Angela, Allegretta Caterina, Pastorino Cristina, Pedemonte Nicoletta, Falchi Federico, Laselva Onofrio, Bandiera Tiziano, Bertozzi Fabio