日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Direct-to-Biology Enabled Molecular Glue Discovery

直接应用于生物学领域的分子胶发现

Hu, Maowei; Ochoada, Jason; Actis, Marisa; McGowan, Kevin; Jarusiewicz, Jamie A; Yoshimura, Satoshi; McGrath, Logan; Neelakantan, Uma; Aggarwal, Anup; Mayasundari, Anand; Young, Sarah M; Zhang, Meng; Yang, Lei; Li, Yong; Mercer, Shea; Babu, M Madan; Fischer, Marcus; Young, Brandon M; Yang, Jun J; Nishiguchi, Gisele; Shelat, Anang A; Blair, Daniel J

BRD4 recruitment desilences transcription without erasure or depletion of repressive chromatin

BRD4 的募集能够解除转录沉默,而无需擦除或耗竭抑制性染色质。

Brandon, Christopher J; Robinson-Thiewes, Sarah; Kaulage, Mangesh; Rosikiewicz, Wojciech; Cuneo, Matthew J; Brett, Joseph; Kandola, Jindpreet; Lang, Walter H; Low, Jonathan; Mohammed, Ashraf; Danda, Adithi; Rider, Sam; Valentine, Marcus; Ochoada, Jason; Young, Brandon; Nguyen, Theresa; Kietlinska, Sandra J; Taylor, Aaron B; Hoeckendorf, Burkhard; Rodrigues, Patrick; Lin, Wenwei; Khairy, Khaled; Xu, Beisi; Shelat, Anang A; Chen, Taosheng; Mittag, Tanja; Ansari, Aseem Z

HTS Identifies NUP98-KDM5A-PHD3 Domain Ligands with Novel Scaffolds

高通量筛选鉴定出具有新型支架的NUP98-KDM5A-PHD3结构域配体

Lin, Wenwei; Slavish, P Jake; Phillips, Aaron H; Trotter, Marlon; Yang, Guangwei; Chai, Sergio C; Churion, Kelly; Ochoada, Jason; Das, Sourav; Shelat, Anang A; Mullighan, Charles G; Kriwacki, Richard W; Rankovic, Zoran; Chen, Taosheng

Principles of paralog-specific targeted protein degradation engaging the C-degron E3 KLHDC2

参与 C-降解决定子 E3 KLHDC2 的同源物特异性靶向蛋白质降解的原理

Daniel C Scott #, Suresh Dharuman #, Elizabeth Griffith, Sergio C Chai, Jarrid Ronnebaum, Moeko T King, Rajendra Tangallapally, Chan Lee, Clifford T Gee, Lei Yang, Yong Li, Victoria C Loudon, Ha Won Lee, Jason Ochoada, Darcie J Miller, Thilina Jayasinghe, Joao A Paulo, Stephen J Elledge, J Wade Harp

Evaluating and evolving a screening library in academia: the St Jude approach

评估和发展学术界的筛查库:圣裘德儿童研究医院的方法

Nishiguchi, Gisele; Das, Sourav; Ochoada, Jason; Long, Heather; Lee, Richard E; Rankovic, Zoran; Shelat, Anang A

Identification of Compounds with pH-Dependent Bactericidal Activity against Mycobacterium tuberculosis

具有抗结核分枝杆菌pH依赖性杀菌活性的化合物的鉴定

Julie Early, Juliane Ollinger, Crystal Darby, Torey Alling, Steven Mullen, Allen Casey, Ben Gold, Jason Ochoada, Todd Wiernicki, Thierry Masquelin, Carl Nathan, Philip A Hipskind, Tanya Parish