日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

2H-Thiazolo[4,5-d][1,2,3]triazole: synthesis, functionalization, and application in scaffold-hopping

2H-噻唑并[4,5-d][1,2,3]三唑:合成、功能化及其在骨架跃迁中的应用

Miyazaki, Ryuya; Takada, Fumito; Kikuchi, Takunari; Oguro, Yuya; Kamata, Makoto; Yukawa, Takafumi; Kato, Kenta; Muto, Kei; Yamaguchi, Junichiro

A novel pyrrolo[3, 2-d]pyrimidine derivative, as a vascular endothelial growth factor receptor and platelet-derived growth factor receptor tyrosine kinase inhibitor, shows potent antitumor activity by suppression of tumor angiogenesis.

一种新型吡咯并[3, 2-d]嘧啶衍生物,作为血管内皮生长因子受体和血小板衍生生长因子受体酪氨酸激酶抑制剂,通过抑制肿瘤血管生成显示出强大的抗肿瘤活性

Awazu Yoshiko, Mizutani Akio, Nagase Yoshinori, Iwata Hidehisa, Oguro Yuya, Miki Hiroshi, Imamura Shinichi, Hori Akira