Conversion of a PROTAC Mutant Huntingtin Degrader into Small-Molecule Hydrophobic Tags Focusing on Drug-like Properties
将PROTAC突变亨廷顿蛋白降解剂转化为小分子疏水标签,重点关注其类药特性。
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.1c00500
Hirai, Keigo; Yamashita, Hiroko; Tomoshige, Shusuke; Mishima, Yugo; Niwa, Tatsuya; Ohgane, Kenji; Ishii, Mayumi; Kanamitsu, Kayoko; Ikemi, Yui; Nakagawa, Shinsaku; Taguchi, Hideki; Sato, Shinichi; Hashimoto, Yuichi; Ishikawa, Minoru