Identification of a Conformational Equilibrium That Determines the Efficacy and Functional Selectivity of the μ-Opioid Receptor
鉴定决定μ-阿片受体效力和功能选择性的构象平衡
期刊:Angewandte Chemie-International Edition
影响因子:16.9
doi:10.1002/anie.201508794
Okude, Junya; Ueda, Takumi; Kofuku, Yutaka; Sato, Motohiko; Nobuyama, Naoyuki; Kondo, Keita; Shiraishi, Yutaro; Mizumura, Takuya; Onishi, Kento; Natsume, Mei; Maeda, Masahiro; Tsujishita, Hideki; Kuranaga, Takefumi; Inoue, Masayuki; Shimada, Ichio