Heteroaryl derivatives of suvorexant as OX1R selective PET ligand candidates: Cu-mediated 18F-fluorination of boroxines, in vitro and initial in vivo evaluation
杂芳基衍生物作为 OX1R 选择性 PET 配体候选物:Cu 介导的硼氧烷 18F 氟化,体外和体内初步评估
期刊:Ejnmmi Research
影响因子:3.1
doi:10.1186/s13550-024-01141-2
Kim-Viktoria Bolik, Jan Hellmann, Simone Maschauer, Eduard Neu, Jürgen Einsiedel, Patrick Riss, Nora Vogg, Jörg König, Martin F Fromm, Harald Hübner, Peter Gmeiner, Olaf Prante