日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Heteroaryl derivatives of suvorexant as OX1R selective PET ligand candidates: Cu-mediated 18F-fluorination of boroxines, in vitro and initial in vivo evaluation

杂芳基衍生物作为 OX1R 选择性 PET 配体候选物:Cu 介导的硼氧烷 18F 氟化,体外和体内初步评估

Kim-Viktoria Bolik, Jan Hellmann, Simone Maschauer, Eduard Neu, Jürgen Einsiedel, Patrick Riss, Nora Vogg, Jörg König, Martin F Fromm, Harald Hübner, Peter Gmeiner, Olaf Prante

In Vitro Assessment of 177Lu-Labeled Trastuzumab-Targeted Mesoporous Carbon@Silica Nanostructure for the Treatment of HER2-Positive Breast Cancer

177Lu 标记曲妥珠单抗靶向介孔碳@二氧化硅纳米结构治疗 HER2 阳性乳腺癌的体外评估

Ayça Tunçel, Simone Maschauer, Olaf Prante, Fatma Yurt

Radiosynthesis and Preclinical Evaluation of 18F-Labeled Estradiol Derivatives with Different Lipophilicity for PET Imaging of Breast Cancer

不同亲脂性的18F标记雌二醇衍生物的放射合成及用于乳腺癌PET显像的临床前评价

Anna Friedel, Olaf Prante, Simone Maschauer

Neurotensin analogs by fluoroglycosylation at Nω-carbamoylated arginines for PET imaging of NTS1-positive tumors

通过 Nω-氨基甲酰化精氨酸进行氟糖基化,制备神经降压素类似物,用于 NTS1 阳性肿瘤的 PET 成像

Lisa Schindler, Katrin Wohlfahrt, Lara Gluhacevic von Krüchten, Olaf Prante, Max Keller, Simone Maschauer

Bivalent ligands promote endosomal trafficking of the dopamine D3 receptor-neurotensin receptor 1 heterodimer

双价配体促进多巴胺 D3 受体-神经降压素受体 1 异二聚体的内体运输

Julian Budzinski, Simone Maschauer, Hiroyuki Kobayashi, Pierre Couvineau, Hannah Vogt, Peter Gmeiner, Anna Roggenhofer, Olaf Prante, Michel Bouvier, Dorothee Weikert

Pharmacological Characterization of Low-to-Moderate Affinity Opioid Receptor Agonists and Brain Imaging with 18F-Labeled Derivatives in Rats

低至中等亲和力阿片受体激动剂的药理学表征及大鼠 18F 标记衍生物的脑成像

Julian Ott, Mona M Spilhaug, Simone Maschauer, Waqas Rafique, Jimmy E Jakobsson, Karoline Hartvig, Harald Hübner, Peter Gmeiner, Olaf Prante, Patrick J Riss

18F-labelled triazolyl-linked argininamides targeting the neuropeptide Y Y1R for PET imaging of mammary carcinoma

18F 标记的三唑基连接精氨酰胺靶向神经肽 Y Y1R 用于乳腺癌的 PET 成像

Simone Maschauer, Julian J Ott, Günther Bernhardt, Torsten Kuwert, Max Keller, Olaf Prante

Theranostic Value of Multimers: Lessons Learned from Trimerization of Neurotensin Receptor Ligands and Other Targeting Vectors

多聚体的治疗诊断价值:从神经降压素受体配体三聚化和其他靶向载体中吸取的经验教训

Simone Maschauer, Jürgen Einsiedel, Dominik Reich, Harald Hübner, Peter Gmeiner, Hans-Jürgen Wester, Olaf Prante, Johannes Notni

In Vitro and In Vivo Characterization of Selected Fluorine-18 Labeled Radioligands for PET Imaging of the Dopamine D3 Receptor

用于多巴胺 D3 受体 PET 成像的氟-18 标记放射性配体的体外和体内表征

Natascha Nebel, Simone Maschauer, Torsten Kuwert, Carsten Hocke, Olaf Prante

H-CRRETAWAC-OH, a lead structure for the development of radiotracer targeting integrin α5β1?

H-CRRETAWAC-OH,是开发针对整合素 α5β1 的放射性示踪剂的先导结构吗?

Roland Haubner, Simone Maschauer, Jürgen Einsiedel, Iris E Eder, Christine Rangger, Peter Gmeiner, Irene J Virgolini, Olaf Prante