日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inhibiting Type I Arginine Methyltransferase Activity Promotes T Cell-Mediated Antitumor Immune Responses

抑制I型精氨酸甲基转移酶活性可促进T细胞介导的抗肿瘤免疫反应

Andrew Fedoriw # ,Leilei Shi # ,Shane O'Brien ,Kimberly N Smitheman ,Yunfei Wang ,Jiakai Hou ,Christian Sherk ,Satyajit Rajapurkar ,Jenny Laraio ,Leila J Williams ,Chunyu Xu ,Guangchun Han ,Qin Feng ,Mark T Bedford ,Linghua Wang ,Olena Barbash ,Ryan G Kruger ,Patrick Hwu ,Helai P Mohammad ,Weiyi Peng

A Chemical Acetylation-Based Mass Spectrometry Platform for Histone Methylation Profiling

基于化学乙酰化的组蛋白甲基化分析质谱平台

Francesca Zappacosta, Craig D Wagner, Anthony Della Pietra 3rd, Sarah V Gerhart, Kathryn Keenan, Susan Korenchuck, Chad J Quinn, Olena Barbash, Michael T McCabe, Roland S Annan

Limited antitumor activity of combined BET and MEK inhibition in neuroblastoma

BET 和 MEK 联合抑制对神经母细胞瘤的抗肿瘤活性有限

Jason R Healy, Lori S Hart, Alexander L Shazad, Maria E Gagliardi, Matthew Tsang, Jimmy Elias, Jacob Ruden, Alvin Farrel, Jo Lynne Rokita, Yimei Li, Anastasia Wyce, Olena Barbash, Vandana Batra, Minu Samanta, John M Maris, Robert W Schnepp

Therapeutic Targeting of RNA Splicing Catalysis through Inhibition of Protein Arginine Methylation

通过抑制蛋白质精氨酸甲基化来靶向RNA剪接催化进行治疗

Jia Yi Fong,Luca Pignata,Pierre-Alexis Goy,Kimihito Cojin Kawabata,Stanley Chun-Wei Lee,Cheryl M Koh,Daniele Musiani,Enrico Massignani,Andriana G Kotini,Alex Penson,Cheng Mun Wun,Yudao Shen,Megan Schwarz,Diana Hp Low,Alexander Rialdi,Michelle Ki,Heike Wollmann,Slim Mzoughi,Florence Gay,Christine Thompson,Timothy Hart,Olena Barbash,Genna M Luciani,Magdalena M Szewczyk,Bas J Wouters,Ruud Delwel,Eirini P Papapetrou,Dalia Barsyte-Lovejoy,Cheryl H Arrowsmith,Mark D Minden,Jian Jin,Ari Melnick,Tiziana Bonaldi,Omar Abdel-Wahab,Ernesto Guccione

Targeting enhancer switching overcomes non-genetic drug resistance in acute myeloid leukaemia

靶向增强子转换可克服急性髓系白血病中的非遗传性耐药性

Charles C Bell ,Katie A Fennell ,Yih-Chih Chan ,Florian Rambow ,Miriam M Yeung ,Dane Vassiliadis ,Luis Lara ,Paul Yeh ,Luciano G Martelotto ,Aljosja Rogiers ,Brandon E Kremer ,Olena Barbash ,Helai P Mohammad ,Timothy M Johanson ,Marian L Burr ,Arindam Dhar ,Natalie Karpinich ,Luyi Tian ,Dean S Tyler ,Laura MacPherson ,Junwei Shi ,Nathan Pinnawala ,Chun Yew Fong ,Anthony T Papenfuss ,Sean M Grimmond ,Sarah-Jane Dawson ,Rhys S Allan ,Ryan G Kruger ,Christopher R Vakoc ,David L Goode ,Shalin H Naik ,Omer Gilan ,Enid Y N Lam ,Jean-Christophe Marine ,Rab K Prinjha ,Mark A Dawson

Activation of the p53-MDM4 regulatory axis defines the anti-tumour response to PRMT5 inhibition through its role in regulating cellular splicing

p53-MDM4 调节轴的激活通过其在调节细胞剪接中的作用决定了对 PRMT5 抑制的抗肿瘤反应

Sarah V Gerhart, Wendy A Kellner, Christine Thompson, Melissa B Pappalardi, Xi-Ping Zhang, Rocio Montes de Oca, Elayne Penebre, Kenneth Duncan, Ann Boriack-Sjodin, BaoChau Le, Christina Majer, Michael T McCabe, Chris Carpenter, Neil Johnson, Ryan G Kruger, Olena Barbash

PRMT5 Is a Critical Regulator of Breast Cancer Stem Cell Function via Histone Methylation and FOXP1 Expression

PRMT5 通过组蛋白甲基化和 FOXP1 表达调节乳腺癌干细胞功能

Kelly Chiang, Agnieszka E Zielinska, Abeer M Shaaban, Maria Pilar Sanchez-Bailon, James Jarrold, Thomas L Clarke, Jingxian Zhang, Adele Francis, Louise J Jones, Sally Smith, Olena Barbash, Ernesto Guccione, Gillian Farnie, Matthew J Smalley, Clare C Davies

SMYD3 links lysine methylation of MAP3K2 to Ras-driven cancer

SMYD3 将 MAP3K2 的赖氨酸甲基化与 Ras 驱动的癌症联系起来

Pawel K Mazur, Nicolas Reynoird, Purvesh Khatri, Pascal W T C Jansen, Alex W Wilkinson, Shichong Liu, Olena Barbash, Glenn S Van Aller, Michael Huddleston, Dashyant Dhanak, Peter J Tummino, Ryan G Kruger, Benjamin A Garcia, Atul J Butte, Michiel Vermeulen, Julien Sage, Or Gozani

Potent antimyeloma activity of the novel bromodomain inhibitors I-BET151 and I-BET762

新型溴结构域抑制剂 I-BET151 和 I-BET762 具有强效抗骨髓瘤活性

Aristeidis Chaidos, Valentina Caputo, Katerina Gouvedenou, Binbin Liu, Ilaria Marigo, Mohammed Suhail Chaudhry, Antonia Rotolo, David F Tough, Nicholas N Smithers, Anna K Bassil, Trevor D Chapman, Nicola R Harker, Olena Barbash, Peter Tummino, Niam Al-Mahdi, Andrea C Haynes, Leanne Cutler, BaoChau L