日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Backbone Alterations in Cyclic Peptides Influence Both Membrane Permeability and Biological Activity

环肽骨架的改变会影响膜通透性和生物活性。

Openy, Joseph; Vega-Ces, Sabela; Amrahova, Gulshan; Mestdach, Emeline; Chi, Celestine; Kissel, Benjamin; 't Hart, Peter

Interplay of Stereochemistry and Charge Governs Guest Binding in Flexible Zn(II)(4)L(4) Cages

立体化学和电荷的相互作用控制着柔性 Zn(II)4L(4) 笼中的客体结合

Xue, Weichao; Benchimol, Elie; Walther, Alexandre; Ouyang, Nianfeng; Holstein, Julian J; Ronson, Tanya K; Openy, Joseph; Zhou, Yujuan; Wu, Kai; Chowdhury, Rituparno; Clever, Guido H; Nitschke, Jonathan R

On-Resin Photochemical Decarboxylative Arylation of Peptides

肽的树脂上光化学脱羧芳基化反应

Pal, Sunit; Openy, Joseph; Krzyzanowski, Adrian; Noisier, Anaïs; 't Hart, Peter

Rationally designed stapled peptides allosterically inhibit PTBP1-RNA-binding

合理设计的环状肽通过变构作用抑制PTBP1-RNA结合

Schmeing, Stefan; Amrahova, Gulshan; Bigler, Katrin; Chang, Jen-Yao; Openy, Joseph; Pal, Sunit; Posada, Laura; Gasper, Raphael; 't Hart, Peter

Solid-Phase Peptide Modification via Deaminative Photochemical Csp(3) -Csp(3) Bond Formation Using Katritzky Salts

利用卡特里茨基盐通过脱氨光化学Csp(3)-Csp(3)键形成进行固相肽修饰

Openy, Joseph; Amrahova, Gulshan; Chang, Jen-Yao; Noisier, Anaïs; Hart, Peter 't

Apparent density, trypanosome infection rates and host preference of tsetse flies in the sleeping sickness endemic focus of northwestern Uganda

乌干达西北部昏睡病流行区采采蝇的表观密度、锥虫感染率和宿主偏好

Opiro, Robert; Opoke, Robert; Angwech, Harriet; Nakafu, Esther; Oloya, Francis A; Openy, Geoffrey; Njahira, Moses; Macharia, Mercy; Echodu, Richard; Malinga, Geoffrey M; Opiyo, Elizabeth A

Antivenin plants used for treatment of snakebites in Uganda: ethnobotanical reports and pharmacological evidences

乌干达用于治疗蛇咬伤的抗蛇毒植物:民族植物学报告和药理学证据

Omara, Timothy; Kagoya, Sarah; Openy, Abraham; Omute, Tom; Ssebulime, Stephen; Kiplagat, Kibet Mohamed; Bongomin, Ocident

Prevalence of diarrhoea and associated risk factors among children under five years old in Pader District, northern Uganda

乌干达北部帕德尔区五岁以下儿童腹泻患病率及相关危险因素

Omona, Stephen; Malinga, Geoffrey M; Opoke, Robert; Openy, Geoffrey; Opiro, Robert

Synthesis and Pharmacological Evaluation of Triazolopyrimidinone Derivatives as Noncompetitive, Intracellular Antagonists for CC Chemokine Receptors 2 and 5

三唑并嘧啶酮衍生物作为 CC 趋化因子受体 2 和 5 的非竞争性细胞内拮抗剂的合成和药理学评价

Natalia V Ortiz Zacarías, Jacobus P D van Veldhoven, Lisa S den Hollander, Burak Dogan, Joseph Openy, Ya-Yun Hsiao, Eelke B Lenselink, Laura H Heitman, Adriaan P IJzerman

Prevalence of lower limb deep venous thrombosis among adult HIV positive patients attending an outpatient clinic at Mulago Hospital

穆拉戈医院门诊就诊的成年HIV阳性患者中下肢深静脉血栓的患病率

Vululi, Sosthene Tsongo; Bugeza, Samuel; Zeridah, Muyinda; Ddungu, Henry; Openy, Akello Betty; Frank, Mubiru; Parkes-Ratanshi, Rosalind