Sulfonyl Anthranilic Acid Analogues Display Pan-Serotype Anti-Dengue Activity by Downregulating the Expression of Ribosomal Proteins Encoded by 5'-Terminal Oligopyrimidine Motif-Containing mRNA
磺酰邻氨基苯甲酸类似物通过下调由含5'末端寡嘧啶基序的mRNA编码的核糖体蛋白的表达,表现出泛血清型抗登革热活性。
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c03414
Gwee, Chin Piaw; Felicetti, Tommaso; Chan, Kitti Wing Ki; Tan, Min Jie Alvin; Bin Mohd Mazlan, Muhammad Danial; Milite, Ciro; Pepe, Giacomo; Sarnari, Chiara; Ng, Xiao Dan; Phoo, Wint Wint; Tan, Jasmine Hwee Yee; Mah, Marcus G; Watanabe, Satoru; Huang, Jing Xiu; Massari, Serena; Tabarrini, Oriana; Sabatini, Stefano; Campiglia, Pietro; Sbardella, Gianluca; Smith, Gavin J D; Alonso, Sylvie; Sun, Alfred Xuyang; Sobota, Radoslaw M; Vasudevan, Subhash G; Manfroni, Giuseppe