日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

AZ14289671 is a highly selective and blood-brain barrier penetrant irreversible TKI that targets EGFRExon20 insertions.

AZ14289671 是一种高选择性且能穿透血脑屏障的不可逆 TKI,靶向 EGFRExon20 插入

Swaih Aisha M, Talbot Sara, Savoca Adriana, Thorpe Hannah, Flemington Vikki, Phillips Benjamin, Colclough Nicola, McCoull William, Radeva Veronika, Hargreaves David, Packer Martin J, Felisberto-Rodrigues Catarina, Thomson Clare, Orme Jonathan P, Deane Carly, Smith Aaron, Johnström Peter, Schou Magnus, McWilliams Lisa, Davey Paul, Enget Marianne, O'Neill Daniel, Cosulich Sabina, Floc'h Nicolas

Vinylpyridine as a Tunable Covalent Warhead Targeting C797 in EGFR.

乙烯基吡啶作为可调控共价弹头靶向 EGFR 中的 C797

Pemberton Nils, Compagne Nina, Argyrou Argyrides, Evertsson Emma, Gunnarsson Anders, Kettle Jason G, Orme Jonathan P, Ward Richard A

Endoproteolytic cleavage of TUG protein regulates GLUT4 glucose transporter translocation

TUG 蛋白的内切蛋白酶切割调节 GLUT4 葡萄糖转运蛋白的转运

Jonathan S Bogan, Bradley R Rubin, Chenfei Yu, Michael G Löffler, Charisse M Orme, Jonathan P Belman, Leah J McNally, Mingming Hao, James A Cresswell