Discovery of EGT710, an Oral Nonpeptidomimetic Reversible Covalent SARS-CoV-2 Main Protease Inhibitor
发现 EGT710，一种口服非肽模拟可逆共价 SARS-CoV-2 主蛋白酶抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c02360
Papillon, Julien P N; Yuan, Jun; Hesse, Matthew J; Zhang, Lei; Robinson, Richard I; Ware, Nathaniel F; Hornak, Viktor; Karki, Rajeshri G; Kirrane, Tom; Garland, Keira; Joseph, Sajan; Moquin, Stephanie A; Lakshminarayana, Suresh B; Tandeske, Laura; Dovala, Dustin; Knapp, Mark; Ornelas, Elizabeth; Fuller, Daniel; Ho, Pei-I; Xie, Xuping; Vulic, Katarina; Skolnik, Suzanne M; Gao, Jinhai; Zambrowski, Mark; Spiess, Meike; Duca, José S; Busby, Scott A; Schirle, Markus; Robinson, Michael; Shi, Pei-Yong; Moser, Heinz E; Sarko, Christopher; Bradner, James E; Diagana, Thierry T; Tallarico, John A
