Apralogs: Apramycin 5-O-Glycosides and Ethers with Improved Antibacterial Activity and Ribosomal Selectivity and Reduced Susceptibility to the Aminoacyltranserferase (3)-IV Resistance Determinant.
Apralogs:Apramycin 5-O-糖苷和醚,具有改进的抗菌活性和核糖体选择性,并降低了对氨酰转移酶(3)-IV 耐药决定簇的敏感性
期刊:Journal of the American Chemical Society
影响因子:15.6
doi:10.1021/jacs.9b11601
Quirke Jonathan C K, Rajasekaran Parasuraman, Sarpe Vikram A, Sonousi Amr, Osinnii Ivan, Gysin Marina, Haldimann Klara, Fang Qiao-Jun, Shcherbakov Dimitri, Hobbie Sven N, Sha Su-Hua, Schacht Jochen, Vasella Andrea, Böttger Erik C, Crich David