日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tsc1 Deletion in Purkinje Neurons Disrupts the Axon Initial Segment, Impairing Excitability and Cerebellar Function

浦肯野神经元中Tsc1基因的缺失会破坏轴突起始段,损害其兴奋性和小脑功能。

Brown, Samuel P; Jena, Achintya K; Osko, Joanna J; Ransdell, Joseph L

Selective deletion of Tsc1 from mouse cerebellar Purkinje neurons drives sex-specific behavioral impairments linked to autism

选择性删除小鼠小脑浦肯野神经元中的Tsc1基因会导致与自闭症相关的性别特异性行为障碍

Lawson, Ryan J; Lipovsek, Nicholas J; Brown, Samuel P; Jena, Achintya K; Osko, Joanna J; Ransdell, Joseph L

Harnessing the Role of HDAC6 in Idiopathic Pulmonary Fibrosis: Design, Synthesis, Structural Analysis, and Biological Evaluation of Potent Inhibitors

利用 HDAC6 在特发性肺纤维化中的作用:强效抑制剂的设计、合成、结构分析和生物学评估

Giuseppe Campiani, Caterina Cavella, Jeremy D Osko, Margherita Brindisi, Nicola Relitti, Simone Brogi, A Prasanth Saraswati, Stefano Federico, Giulia Chemi, Samuele Maramai, Gabriele Carullo, Benedikt Jaeger, Alfonso Carleo, Rosaria Benedetti, Federica Sarno, Stefania Lamponi, Paola Rottoli, Elena B

Structural analysis of histone deacetylase 8 mutants associated with Cornelia de Lange Syndrome spectrum disorders

与 Cornelia de Lange 综合征谱系障碍相关的组蛋白去乙酰化酶 8 突变体的结构分析

Jeremy D Osko, Nicholas J Porter, Christophe Decroos, Matthew S Lee, Paris R Watson, Sarah E Raible, Ian D Krantz, Matthew A Deardorff, David W Christianson

Multicomponent Synthesis, Binding Mode, and Structure-Activity Relationship of Selective Histone Deacetylase 6 (HDAC6) Inhibitors with Bifurcated Capping Groups

具有双分支封端基团的选择性组蛋白去乙酰化酶 6 (HDAC6) 抑制剂的多组分合成、结合模式及构效关系

Nina Reßing, Melf Sönnichsen, Jeremy D Osko, Andrea Schöler, Julian Schliehe-Diecks, Alexander Skerhut, Arndt Borkhardt, Julia Hauer, Matthias U Kassack, David W Christianson, Sanil Bhatia, Finn K Hansen

Spiroindoline-Capped Selective HDAC6 Inhibitors: Design, Synthesis, Structural Analysis, and Biological Evaluation

螺吲哚啉封端的选择性HDAC6抑制剂:设计、合成、结构分析和生物学评价

Saraswati, A Prasanth; Relitti, Nicola; Brindisi, Margherita; Osko, Jeremy D; Chemi, Giulia; Federico, Stefano; Grillo, Alessandro; Brogi, Simone; McCabe, Niamh H; Turkington, Richard C; Ibrahim, Ola; O'Sullivan, Jeffrey; Lamponi, Stefania; Ghanim, Magda; Kelly, Vincent P; Zisterer, Daniela; Amet, Rebecca; Hannon Barroeta, Patricia; Vanni, Francesca; Ulivieri, Cristina; Herp, Daniel; Sarno, Federica; Di Costanzo, Antonella; Saccoccia, Fulvio; Ruberti, Giovina; Jung, Manfred; Altucci, Lucia; Gemma, Sandra; Butini, Stefania; Christianson, David W; Campiani, Giuseppe

Design and Synthesis of Dihydroxamic Acids as HDAC6/8/10 Inhibitors

二羟肟酸作为 HDAC6/8/10 抑制剂的设计和合成

Michael Morgen, Raphael R Steimbach, Magalie Géraldy, Lars Hellweg, Peter Sehr, Johannes Ridinger, Olaf Witt, Ina Oehme, Corey J Herbst-Gervasoni, Jeremy D Osko, Nicholas J Porter, David W Christianson, Nikolas Gunkel, Aubry K Miller

Eurados review of retrospective dosimetry techniques for internal exposures to ionising radiation and their applications

欧洲辐射防护协会(Eurados)对电离辐射内照射回顾性剂量测定技术及其应用的审查

Giussani, A; Lopez, M A; Romm, H; Testa, A; Ainsbury, E A; Degteva, M; Della Monaca, S; Etherington, G; Fattibene, P; Güclu, I; Jaworska, A; Lloyd, D C; Malátová, I; McComish, S; Melo, D; Osko, J; Rojo, A; Roch-Lefevre, S; Roy, L; Shishkina, E; Sotnik, N; Tolmachev, S Y; Wieser, A; Woda, C; Youngman, M

Structural determinants of affinity and selectivity in the binding of inhibitors to histone deacetylase 6

抑制剂与组蛋白去乙酰化酶6结合的亲和力和选择性的结构决定因素

Osko, Jeremy D; Christianson, David W

Binding of inhibitors to active-site mutants of CD1, the enigmatic catalytic domain of histone deacetylase 6

抑制剂与组蛋白去乙酰化酶6的神秘催化结构域CD1活性位点突变体的结合

Osko, Jeremy D; Christianson, David W