日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Human acid-sensing ion channel 1a/3 heteromers at a 1:2 ratio expand the functional capabilities of homomeric ASIC3 and are likely to be physiologically relevant

人类酸敏感离子通道 1a/3 异源二聚体以 1:2 的比例形成,扩展了同源二聚体 ASIC3 的功能,并可能具有生理相关性。

Osmakov, Dmitry I; Dubodel, Elisaveta S; Kalinovskii, Aleksandr P; Koshelev, Sergey G; Andreev, Yaroslav A; Korolkova, Yuliya V; Kozlov, Sergey A

Two Amino Acid Substitutions Improve the Pharmacological Profile of the Snake Venom Peptide Mambalgin

两种氨基酸取代改善了蛇毒肽马巴尔金的药理学特性

Osmakov, Dmitry I; Khasanov, Timur A; Maleeva, Ekaterina E; Pavlov, Vladimir M; Palikov, Victor A; Belozerova, Olga A; Koshelev, Sergey G; Korolkova, Yuliya V; Dyachenko, Igor A; Kozlov, Sergey A; Andreev, Yaroslav A

Opioid Analgesic as a Positive Allosteric Modulator of Acid-Sensing Ion Channels

阿片类镇痛药作为酸敏感离子通道的正向变构调节剂

Osmakov, Dmitry I; Onoprienko, Lyudmila V; Kalinovskii, Aleksandr P; Koshelev, Sergey G; Stepanenko, Vasiliy N; Andreev, Yaroslav A; Kozlov, Sergey A

Dual Modulator of ASIC Channels and GABA(A) Receptors from Thyme Alters Fear-Related Hippocampal Activity

百里香来源的ASIC通道和GABA(A)受体双重调节剂改变与恐惧相关的海马活动

Kalinovskii, Aleksandr P; Pushkarev, Anton P; Mikhailenko, Anastasia D; Kudryavtsev, Denis S; Belozerova, Olga A; Shmygarev, Vladimir I; Yatskin, Oleg N; Korolkova, Yuliya V; Kozlov, Sergey A; Osmakov, Dmitry I; Popov, Alexander; Andreev, Yaroslav A

Anxiolytic, Analgesic and Anti-Inflammatory Effects of Peptides Hmg 1b-2 and Hmg 1b-4 from the Sea Anemone Heteractis magnifica

海葵 Heteractis magnifica 中的肽 Hmg 1b-2 和 Hmg 1b-4 具有抗焦虑、镇痛和抗炎作用

Irina N Gladkikh, Anna A Klimovich, Rimma S Kalina, Yulia V Kozhevnikova, Timur A Khasanov, Dmitry I Osmakov, Sergey G Koshelev, Margarita M Monastyrnaya, Yaroslav A Andreev, Elena V Leychenko, Sergey A Kozlov

Lignans as Pharmacological Agents in Disorders Related to Oxidative Stress and Inflammation: Chemical Synthesis Approaches and Biological Activities

木脂素作为氧化应激和炎症相关疾病的药理活性物质:化学合成方法和生物活性

Osmakov, Dmitry I; Kalinovskii, Aleksandr P; Belozerova, Olga A; Andreev, Yaroslav A; Kozlov, Sergey A

Retinoic Acid-Differentiated Neuroblastoma SH-SY5Y Is an Accessible In Vitro Model to Study Native Human Acid-Sensing Ion Channels 1a (ASIC1a)

视黄酸分化神经母细胞瘤 SH-SY5Y 是一种可用于研究天然人类酸敏感离子通道 1a (ASIC1a) 的体外模型

Kalinovskii, Aleksandr P; Osmakov, Dmitry I; Koshelev, Sergey G; Lubova, Kseniya I; Korolkova, Yuliya V; Kozlov, Sergey A; Andreev, Yaroslav A

Animal, Herb, and Microbial Toxins for Structural and Pharmacological Study of Acid-Sensing Ion Channels

用于酸敏感离子通道结构和药理学研究的动物、草药和微生物毒素

Osmakov, Dmitry I; Khasanov, Timur A; Andreev, Yaroslav A; Lyukmanova, Ekaterina N; Kozlov, Sergey A

Mambalgin-2 Induces Cell Cycle Arrest and Apoptosis in Glioma Cells via Interaction with ASIC1a

Mambalgin-2 通过与 ASIC1a 相互作用诱导胶质瘤细胞周期停滞和凋亡

Maxim Bychkov, Mikhail Shulepko, Dmitry Osmakov, Yaroslav Andreev, Anastasia Sudarikova, Valeria Vasileva, Marat S Pavlyukov, Yaroslav A Latyshev, Alexander A Potapov, Mikhail Kirpichnikov, Zakhar O Shenkarev, Ekaterina Lyukmanova

Endogenous Neuropeptide Nocistatin Is a Direct Agonist of Acid-Sensing Ion Channels (ASIC1, ASIC2 and ASIC3)

内源性神经肽 Nocistatin 是酸敏感离子通道 (ASIC1、ASIC2 和 ASIC3) 的直接激动剂

Dmitry I Osmakov, Sergey G Koshelev, Igor A Ivanov, Yaroslav A Andreev, Sergey A Kozlov