日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Therapeutic potential of allosteric HECT E3 ligase inhibition.

变构 HECT E3 连接酶抑制的治疗潜力

Rothman Alexander M K, Florentin Amir, Zink Florence, Quigley Catherine, Bonneau Olivier, Hemmig Rene, Hachey Amanda, Rejtar Tomas, Thaker Maulik, Jain Rishi, Huang Shih-Min, Sutton Daniel, Roger Jan, Zhang Ji-Hu, Weiler Sven, Cotesta Simona, Ottl Johannes, Srivastava Salil, Kordonsky Alina, Avishid Reut, Yariv Elon, Rathi Ritu, Khvalevsky Oshrit, Troxler Thomas, Binmahfooz Sarah K, Kleifeld Oded, Morrell Nicholas W, Humbert Marc, Thomas Matthew J, Jarai Gabor, Beckwith Rohan E J, Cobb Jennifer S, Smith Nichola, Ostermann Nils, Tallarico John, Shaw Duncan, Guth-Gundel Sabine, Prag Gali, Rowlands David J

Identification and characterization of binders to a cryptic and functional pocket in KRAS

鉴定和表征KRAS中隐蔽功能口袋的结合蛋白

Beyer, Kim S; Klein, Jessica; Katz, Stéphanie; Welker, Patrick; Lanter, Mylene; Guthy, Daniel; Pollehn, Kerstin; Gluck-Gadé, Aurélie; Bleu, Melusine; Desogus, Jessica; Hattenberger, Marc; Borrello, Damiano; Abdul Rahman, Wassim; Zink, Florence; Ostermann, Nils; Jahnke, Wolfgang; Dumelin, Christoph E; Leder, Lukas; Esser, Oliver; Muller, Lionel; Marzinzik, Andreas; Cébé, Regis; Müller, Kathrin; Galli, Giorgio G; Tordella, Luca; Cotesta, Simona; Brachmann, Saskia M; Maira, Sauveur-Michel

Oxidatively Induced Reductive N(2) Binding: A Dinickel-Bridging Bent N(2) Radical Anion and Its Redox-Triggered N(2) Release

氧化诱导的还原性N₂结合:双镍桥联弯曲N₂自由基阴离子及其氧化还原触发的N₂释放

Mozzi, Sara I; Manz, Dennis-Helmut; Ostermann, Nils; Schulz, Roland A; Duan, Peng-Cheng; Kothe, Thomas; Diefenbach, Martin; Dechert, Sebastian; Demeshko, Serhiy; Krewald, Vera; Siewert, Inke; Meyer, Franc

Mechanistic Studies of the Proton-Coupled Electron Transfer Reactivity of a Cobalt Complex with a Proton-Responsive PNP Pincer-Type Ligand

质子响应型PNP钳形配体与钴配合物的质子耦合电子转移反应机理研究

Mukherjee, Jyotima; Ostermann, Nils; Pecak, Jan; Otte, Matthias; Podewitz, Maren; Siewert, Inke

Dynamic conformational equilibria in the active states of KRAS and NRAS

KRAS和NRAS活性状态下的动态构象平衡

Rennella, Enrico; Henry, Chrystèle; Dickson, Callum J; Georgescauld, Florian; Wales, Thomas E; Erdmann, Dirk; Cotesta, Simona; Maira, Michel; Sedrani, Richard; Brachmann, Saskia M; Ostermann, Nils; Engen, John R; Kay, Lewis E; Beyer, Kim S; Wilcken, Rainer; Jahnke, Wolfgang

(Electro)chemical N2 Splitting by a Molybdenum Complex with an Anionic PNP Pincer-Type Ligand

阴离子 PNP 钳型配体的钼配合物进行(电)化学 N2 裂解

Nils Ostermann, Nils Rotthowe, A Claudia Stückl, Inke Siewert

Structure-based design of substituted piperidines as a new class of highly efficacious oral direct Renin inhibitors

基于结构的取代哌啶类化合物设计作为一类新型高效口服直接肾素抑制剂

Ehara, Takeru; Irie, Osamu; Kosaka, Takatoshi; Kanazawa, Takanori; Breitenstein, Werner; Grosche, Philipp; Ostermann, Nils; Suzuki, Masaki; Kawakami, Shimpei; Konishi, Kazuhide; Hitomi, Yuko; Toyao, Atsushi; Gunji, Hiroki; Cumin, Frederic; Schiering, Nikolaus; Wagner, Trixie; Rigel, Dean F; Webb, Randy L; Maibaum, Jürgen; Yokokawa, Fumiaki