日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inhibition of triple negative breast cancer-associated inflammation, tumor growth and brain colonization by targeting monoacylglycerol lipase

通过靶向单酰甘油脂肪酶抑制三阴性乳腺癌相关炎症、肿瘤生长和脑定植

Othman Benchama, Sergiy Tyukhtenko, Michael S Malamas, Mark K Williams, Alexandros Makriyannis, Hava Karsenty Avraham

Inhibition of triple negative breast cancer-associated inflammation and progression by N- acylethanolamine acid amide hydrolase (NAAA)

N-酰基乙醇胺酰胺水解酶(NAAA)抑制三阴性乳腺癌相关炎症和进展

Othman Benchama, Michael S Malamas, Kulkarni Praveen, Elizabeth C Ethier, Mark K Williams, Alexandros Makriyannis, Hava Karsenty Avraham

Activation and Signaling Mechanism Revealed by Cannabinoid Receptor-Gi Complex Structures

大麻素受体-Gi复合物结构揭示的激活和信号传导机制

Tian Hua, Xiaoting Li, Lijie Wu, Christos Iliopoulos-Tsoutsouvas, Yuxia Wang, Meng Wu, Ling Shen, Christina A Brust, Spyros P Nikas, Feng Song, Xiyong Song, Shuguang Yuan, Qianqian Sun, Yiran Wu, Shan Jiang, Travis W Grim, Othman Benchama, Edward L Stahl, Nikolai Zvonok, Suwen Zhao, Laura M Bohn, Al

Crystal Structure of the Human Cannabinoid Receptor CB2

人类大麻素受体 CB2 的晶体结构

Xiaoting Li, Tian Hua, Kiran Vemuri, Jo-Hao Ho, Yiran Wu, Lijie Wu, Petr Popov, Othman Benchama, Nikolai Zvonok, K'ara Locke, Lu Qu, Gye Won Han, Malliga R Iyer, Resat Cinar, Nathan J Coffey, Jingjing Wang, Meng Wu, Vsevolod Katritch, Suwen Zhao, George Kunos, Laura M Bohn, Alexandros Makriyannis, R

Novel C-Ring-Hydroxy-Substituted Controlled Deactivation Cannabinergic Analogues

新型 C 环羟基取代的可控失活大麻素类似物

Shashank Kulkarni, Spyros P Nikas, Rishi Sharma, Shan Jiang, Carol A Paronis, Michael Z Leonard, Bin Zhang, Chandrashekhar Honrao, Srikrishnan Mallipeddi, Jimit Girish Raghav, Othman Benchama, Torbjörn U C Järbe, Jack Bergman, Alexandros Makriyannis

A comparison of novel, selective fatty acid amide hydrolase (FAAH), monoacyglycerol lipase (MAGL) or dual FAAH/MAGL inhibitors to suppress acute and anticipatory nausea in rat models

新型选择性脂肪酸酰胺水解酶 (FAAH)、单酰甘油脂肪酶 (MAGL) 或双重 FAAH/MAGL 抑制剂对大鼠模型中急性和预期性恶心的抑制效果比较

Linda A Parker, Cheryl L Limebeer, Erin M Rock, Martin A Sticht, Jordan Ward, Greig Turvey, Othman Benchama, Girija Rajarshi, JodiAnne T Wood, Shakiru O Alapafuja, Alexandros Makriyannis

Controlled-deactivation cannabinergic ligands

控制失活大麻素能配体

Rishi Sharma, Spyros P Nikas, Carol A Paronis, Jodianne T Wood, Aneetha Halikhedkar, Jason Jianxin Guo, Ganesh A Thakur, Shashank Kulkarni, Othman Benchama, Jimit Girish Raghav, Roger S Gifford, Torbjörn U C Järbe, Jack Bergman, Alexandros Makriyannis