日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Leveraging Targeted Protein Degradation for G Protein-Coupled Receptors: The Development of CCR2 Molecular Degraders

利用靶向蛋白降解技术调控G蛋白偶联受体:CCR2分子降解剂的开发

Essa, Khaled; Ortiz Zacarías, Natalia V; Roth, Sascha; Xin, Bo-Tao; de Winter, Sabine; van der Horst, Cas; Bleijs, Bente; de Heiden, Richard A; Voulgaraki, Rodanthi; Neubert, Elsa; Ovaa, Huib; Danen, Erik H J; Mulder, Monique P C; Moreau, Kevin; van der Es, Daan; Heitman, Laura H

USP16 is an ISG15 cross-reactive deubiquitinase that targets pro-ISG15 and ISGylated proteins involved in metabolism

USP16 是一种 ISG15 交叉反应性去泛素化酶,靶向参与代谢的 pro-ISG15 和 ISGylated 蛋白。

Gan, Jin; Pinto-Fernández, Adán; Flierman, Dennis; Akkermans, Jimmy J L L; O'Brien, Darragh P; Greenwood, Helene; Scott, Hannah Claire; Fritz, Günter; Knobeloch, Klaus-Peter; Neefjes, Jacques; van Dam, Hans; Ovaa, Huib; Ploegh, Hidde L; Kessler, Benedikt M; Geurink, Paul P; Sapmaz, Aysegul

In-Plate Chemical Synthesis of Isopeptide-Linked SUMOylated Peptide Fluorescence Polarization Reagents for High-Throughput Screening of SENP Preferences

用于高通量筛选SENP偏好性的异肽连接SUMO化肽荧光偏振试剂的板内化学合成

Huppelschoten, Yara; Mukhopadhyay, Rishov; Buchardt, Jens; Nielsen, Thomas E; Vertegaal, Alfred C O; Ovaa, Huib; van der Heden van Noort, Gerbrand J

Total Chemical Synthesis of a Functionalized GFP Nanobody

功能化GFP纳米抗体的全化学合成

Huppelschoten, Yara; Elhebieshy, Angela F; Hameed, Dharjath S; Sapmaz, Aysegul; Buchardt, Jens; Nielsen, Thomas E; Ovaa, Huib; van der Heden van Noort, Gerbrand J

Ubiquitin ligation to F-box protein targets by SCF-RBR E3-E3 super-assembly

SCF-RBR E3-E3 超组装介导的泛素与 F-box 蛋白靶标的连接

Horn-Ghetko, Daniel; Krist, David T; Prabu, J Rajan; Baek, Kheewoong; Mulder, Monique P C; Klügel, Maren; Scott, Daniel C; Ovaa, Huib; Kleiger, Gary; Schulman, Brenda A

Quantifying Positional Isomers (QPI) by Top-Down Mass Spectrometry

利用自上而下质谱法定量位置异构体(QPI)

Brunner, Andrea M; Lössl, Philip; Geurink, Paul P; Ovaa, Huib; Albanese, P; Altelaar, A F Maarten; Heck, Albert J R; Scheltema, Richard A

Signal inhibitory receptor on leukocytes-1 recognizes bacterial and endogenous amphipathic α-helical peptides.

白细胞上的信号抑制受体-1 可识别细菌和内源性两亲性α螺旋肽

Rumpret Matevž, von Richthofen Helen J, van der Linden Maarten, Westerlaken Geertje H A, Talavera Ormeño Cami, van Strijp Jos A G, Landau Meytal, Ovaa Huib, van Sorge Nina M, Meyaard Linde

Recognition of S100 proteins by Signal Inhibitory Receptor on Leukocytes-1 negatively regulates human neutrophils

白细胞信号抑制受体-1对S100蛋白的识别负向调节人类中性粒细胞

Rumpret, Matevž; von Richthofen, Helen J; van der Linden, Maarten; Westerlaken, Geertje H A; Talavera Ormeño, Cami; Low, Teck Y; Ovaa, Huib; Meyaard, Linde

Targeting TRIM Proteins: A Quest towards Drugging an Emerging Protein Class

靶向TRIM蛋白:探索药物研发新兴蛋白类别

D'Amico, Francesca; Mukhopadhyay, Rishov; Ovaa, Huib; Mulder, Monique P C

Development of Tyrphostin Analogues to Study Inhibition of the Mycobacterium tuberculosis Pup Proteasome System*

开发酪氨酸激酶抑制剂类似物以研究结核分枝杆菌 Pup 蛋白酶体系统的抑制作用*

Janssen, Guido V; Zhang, Susan; Merkx, Remco; Schiesswohl, Christa; Chatterjee, Champak; Darwin, K Heran; Geurink, Paul P; van der Heden van Noort, Gerbrand J; Ovaa, Huib