日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oseltamivir aziridines are potent influenza neuraminidase inhibitors and imaging agents

奥司他韦氮丙啶类药物是强效的流感神经氨酸酶抑制剂和显像剂。

Vriends, Merijn B L; Moran, Elisha; Calvelo, Martín; Hansen, Thomas; Pickles, Isabelle B; Xin, Xincheng; Biezeno, Marieke; Armstrong, Zachary W B; Ferraz, Maria J; Li, Lei; Lilley, Alice; Harvey, Ruth; Filippov, Dmitri V; Liao, Qinghua; Schröder, Sybrin P; van der Marel, Gijsbert A; Artola, Marta; Aerts, Johannes M F G; Blaza, James N; Codée, Jeroen D C; Rovira, Carme; Overkleeft, Herman S; Davies, Gideon J

Fully protected pyrophosphates via phosphorobromidates for the synthesis of biopolymers

利用溴化磷对焦磷酸盐进行完全保护,用于合成生物聚合物

Wijngaarden, Sven; van der Heijden, Femke L A M; Rijpkema, Koen J; van Puffelen, Bob; Meeuwenoord, Nico J; Ramcharan, Danicia; van der Marel, Gijsbert A; Codée, Jeroen D C; Overkleeft, Herman S; Filippov, Dmitri V

Synthesis, Conformal Analysis, and Antibody Binding of Staphylococcus aureus Capsular Polysaccharide Type 5 Oligosaccharides

金黄色葡萄球菌荚膜多糖5型寡糖的合成、保形分析和抗体结合

Østerlid, Kitt E; Li, Sizhe; Unione, Luca; Bino, Linda Del; Sorieul, Charlotte; Carboni, Filippo; Berni, Francesca; Bertuzzi, Sara; van Puffelen, Bob; Arda, Ana; Overkleeft, Herman S; van der Marel, Gijsbert A; Romano, Maria Rosaria; Jiménez-Barbero, Jesús; Adamo, Roberto; Codée, Jeroen D C

Manipulating anthracyclines for deeper tissue penetration and implications for glycolytic tissues

调控蒽环类药物以增强其组织渗透性及其对糖酵解组织的影响

Abels, Erik R; Ter Linden, Esther; Rohling, Jos H T; Voortman, Lennard M; Janssen, Lennert; Hornsveld, Marten; Overkleeft, Herman S; van der Zanden, Sabina Y; Broekman, Marike L D; Neefjes, Jacques

Carfilzomib-specific proteasome β5/β2 inhibition drives cardiotoxicity via remodeling of protein homeostasis and the renin-angiotensin-system

卡非佐米特异性抑制蛋白酶体β5/β2通过重塑蛋白质稳态和肾素-血管紧张素系统而导致心脏毒性。

Max Mendez-Lopez ,Andrej Besse ,Christian Zuppinger ,Christian Perez-Shibayama ,Cristina Gil-Cruz ,Bogdan I Florea ,Angelina De Martin ,Mechthild Lütge ,Deborah Beckerova ,Simon Klimovic ,Xiang Zhou ,Leo Rasche ,Jan Pribyl ,Vladimir Rotrekl ,Burkhard Ludewig ,Herman S Overkleeft ,Lenka Besse ,Christoph Driessen

Inhibitors of the 20S proteasome β5 subunit as potent and selective agents against Trichomonas vaginalis

20S蛋白酶体β5亚基抑制剂作为对抗阴道毛滴虫的有效且选择性药物

Miyamoto, Yukiko; Hurysz, Brianna M; Fajtova, Pavla; Eckmann, Peter; Serafim, Mateus Sá Magalhães; Kronenberger, Thales; Al-Hindy, Momen; Dekker, Patrick M; Maurits, Elmer; Overkleeft, Herman S; Bergdahl, B Mikael; Almaliti, Jehad; Gerwick, William H; O'Donoghue, Anthony J; Eckmann, Lars

Activity-based probes for dynamic characterisation of polysaccharide-degrading enzymes

用于动态表征多糖降解酶的活性探针

Pickles, Isabelle B; Corrêa, Thamy L R; Overkleeft, Herman S; Davies, Gideon J

Activity-Based Protein Profiling Identifies an α-Amylase Family Protein Contributing to the Virulence of Methicillin-Resistant Staphylococcus aureus.

基于活性的蛋白质谱分析鉴定出一种α-淀粉酶家族蛋白,该蛋白有助于耐甲氧西林金黄色葡萄球菌的毒力。

Uddin Md Jalal, Julin Kjersti, Overkleeft Herman S, Johannessen Mona, Lentz Christian S

Convergent Approach Toward ADP-Ribosylated Peptides via a Chemoselective Phosphate Condensation

通过化学选择性磷酸缩合反应合成ADP-核糖基化肽的汇聚方法

Wijngaarden, Sven; van der Heijden, Femke L A M; Bogaart, Cindy J; Siskou, Maria; Tsoumani, Ioanna; Robinson, Daisy J; van der Marel, Gijsbert A; Codée, Jeroen D C; Overkleeft, Herman S; Filippov, Dmitri V

Human milk oligosaccharide 2'-fucosyllactose protects against high-fat diet-induced obesity by changing intestinal mucus production, composition and degradation linked to changes in gut microbiota and faecal proteome profiles in mice

人乳寡糖2'-岩藻糖基乳糖通过改变肠道黏液的产生、组成和降解,进而影响小鼠肠道菌群和粪便蛋白质组的变化,从而起到预防高脂饮食诱导的肥胖的作用。

Paone, Paola; Latousakis, Dimitris; Terrasi, Romano; Vertommen, Didier; Jian, Ching; Borlandelli, Valentina; Suriano, Francesco; Johansson, Malin E V; Puel, Anthony; Bouzin, Caroline; Delzenne, Nathalie M; Salonen, Anne; Juge, Nathalie; Florea, Bogdan I; Muccioli, Giulio G; Overkleeft, Herman; Van Hul, Matthias; Cani, Patrice D