日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oseltamivir aziridines are potent influenza neuraminidase inhibitors and imaging agents

奥司他韦氮丙啶类药物是强效的流感神经氨酸酶抑制剂和显像剂。

Vriends, Merijn B L; Moran, Elisha; Calvelo, Martín; Hansen, Thomas; Pickles, Isabelle B; Xin, Xincheng; Biezeno, Marieke; Armstrong, Zachary W B; Ferraz, Maria J; Li, Lei; Lilley, Alice; Harvey, Ruth; Filippov, Dmitri V; Liao, Qinghua; Schröder, Sybrin P; van der Marel, Gijsbert A; Artola, Marta; Aerts, Johannes M F G; Blaza, James N; Codée, Jeroen D C; Rovira, Carme; Overkleeft, Herman S; Davies, Gideon J

Fully protected pyrophosphates via phosphorobromidates for the synthesis of biopolymers

利用溴化磷对焦磷酸盐进行完全保护,用于合成生物聚合物

Wijngaarden, Sven; van der Heijden, Femke L A M; Rijpkema, Koen J; van Puffelen, Bob; Meeuwenoord, Nico J; Ramcharan, Danicia; van der Marel, Gijsbert A; Codée, Jeroen D C; Overkleeft, Herman S; Filippov, Dmitri V

Synthesis, Conformal Analysis, and Antibody Binding of Staphylococcus aureus Capsular Polysaccharide Type 5 Oligosaccharides

金黄色葡萄球菌荚膜多糖5型寡糖的合成、保形分析和抗体结合

Østerlid, Kitt E; Li, Sizhe; Unione, Luca; Bino, Linda Del; Sorieul, Charlotte; Carboni, Filippo; Berni, Francesca; Bertuzzi, Sara; van Puffelen, Bob; Arda, Ana; Overkleeft, Herman S; van der Marel, Gijsbert A; Romano, Maria Rosaria; Jiménez-Barbero, Jesús; Adamo, Roberto; Codée, Jeroen D C

Long, Synthetic Staphylococcus aureus Type 8 Capsular Oligosaccharides Reveal Structural Epitopes for Effective Immune Recognition

长链合成金黄色葡萄球菌8型荚膜寡糖揭示了有效免疫识别的结构表位

Østerlid, Kitt Emilie; Sorieul, Charlotte; Unione, Luca; Li, Sizhe; García-Sepúlveda, Cristian; Carboni, Filippo; Del Bino, Linda; Berni, Francesca; Arda, Ana; Overkleeft, Herman S; van der Marel, Gijsbert A; Romano, Maria Rosaria; Jiménez-Barbero, Jesús; Adamo, Roberto; Codée, Jeroen D C

Bespoke Activity-Based Probes Reveal that the Pseudomonas aeruginosa Endoglycosidase, PslG, Is an Endo-β-glucanase

定制的活性探针揭示铜绿假单胞菌内切糖苷酶 PslG 是一种内切β-葡聚糖酶

Ruijgrok, Gijs; Offen, Wendy A; Pickles, Isabelle B; Raju, Deepa; Patsos, Thanasis; de Boer, Casper; Ofman, Tim; Rompa, Joep; van Oord, Daan; Dodson, Eleanor J; Beekers, Alexander; Voskuilen, Thijs; Ferrari, Michela; Wu, Liang; Janssen, Antonius P A; Codée, Jeroen D C; Howell, P Lynne; Davies, Gideon J; Overkleeft, Herman S

Manipulating anthracyclines for deeper tissue penetration and implications for glycolytic tissues

调控蒽环类药物以增强其组织渗透性及其对糖酵解组织的影响

Abels, Erik R; Ter Linden, Esther; Rohling, Jos H T; Voortman, Lennard M; Janssen, Lennert; Hornsveld, Marten; Overkleeft, Herman S; van der Zanden, Sabina Y; Broekman, Marike L D; Neefjes, Jacques

Inhibitors of the 20S proteasome β5 subunit as potent and selective agents against Trichomonas vaginalis

20S蛋白酶体β5亚基抑制剂作为对抗阴道毛滴虫的有效且选择性药物

Miyamoto, Yukiko; Hurysz, Brianna M; Fajtova, Pavla; Eckmann, Peter; Serafim, Mateus Sá Magalhães; Kronenberger, Thales; Al-Hindy, Momen; Dekker, Patrick M; Maurits, Elmer; Overkleeft, Herman S; Bergdahl, B Mikael; Almaliti, Jehad; Gerwick, William H; O'Donoghue, Anthony J; Eckmann, Lars

Activity-based probes for dynamic characterisation of polysaccharide-degrading enzymes

用于动态表征多糖降解酶的活性探针

Pickles, Isabelle B; Corrêa, Thamy L R; Overkleeft, Herman S; Davies, Gideon J

Activity-Based Protein Profiling Identifies an α-Amylase Family Protein Contributing to the Virulence of Methicillin-Resistant Staphylococcus aureus.

基于活性的蛋白质谱分析鉴定出一种α-淀粉酶家族蛋白,该蛋白有助于耐甲氧西林金黄色葡萄球菌的毒力。

Uddin Md Jalal, Julin Kjersti, Overkleeft Herman S, Johannessen Mona, Lentz Christian S

Synthesis of a Set of Staphylococcus Aureus Capsular Polysaccharide Type 1 Oligosaccharides Carrying Taurine Esters

合成一组含有牛磺酸酯的金黄色葡萄球菌荚膜多糖I型寡糖

Østerlid, Kitt Emilie; Cergano, Renata; Overkleeft, Herman S; van der Marel, Gijsbert A; Codée, Jeroen D C