Orally Bioavailable BRD4 BD1 Inhibitor ZL0516 Effectively Suppresses Colonic Inflammation in Animal Models of Inflammatory Bowel Disease
口服生物利用度高的BRD4 BD1抑制剂ZL0516可有效抑制炎症性肠病动物模型中的结肠炎症
期刊:ACS Pharmacology and Translational Science
影响因子:3.7
doi:10.1021/acsptsci.5c00068
Ma, Zonghui; McAninch, Steven; Liu, Zhiqing; Zhang, Cun; Chen, Haiying; He, Jing; Yang, Wenjing; Panganiban, Ronaldo P; Cong, Yingzi; Yochum, Gregory; Brasier, Allan R; Pinchuk, Irina V; Tian, Bing; Zhou, Jia
炎症
肠炎
炎症/感染
BRD4
Immunology/Inflammation
结肠炎