日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Activity Relationship of Novel and Selective Biaryl-Chroman GPR40 AgoPAMs

新型选择性联芳基-色满 GPR40 AgoPAMs 的构效关系

Chen, Helen Y; Plummer, Christopher W; Xiao, Dong; Chobanian, Harry R; DeMong, Duane; Miller, Michael; Trujillo, Maria E; Kirkland, Melissa; Kosinski, Daniel; Mane, Joel; Pachanski, Michele; Cheewatrakoolpong, Boonlert; Di Salvo, Jerry; Thomas-Fowlkes, Brande; Souza, Sarah; Tatosian, Daniel A; Chen, Qing; Hafey, Michael J; Houle, Robert; Nolting, Andrew F; Orr, Robert; Ehrhart, Juliann; Weinglass, Adam B; Tschirret-Guth, Richard; Howard, Andrew D; Colletti, Steven L

Discovery of Chromane Propionic Acid Analogues as Selective Agonists of GPR120 with in Vivo Activity in Rodents

发现色满丙酸类似物作为GPR120选择性激动剂,并在啮齿动物体内具有活性

Adams, Gregory L; Velazquez, Francisco; Jayne, Charles; Shah, Unmesh; Miao, Shouwu; Ashley, Eric R; Madeira, Maria; Akiyama, Taro E; Di Salvo, Jerry; Suzuki, Takao; Wang, Nengxue; Truong, Quang; Gilbert, Eric; Zhou, Dan; Verras, Andreas; Kirkland, Melissa; Pachanski, Michele; Powles, Maryann; Yin, Wu; Ujjainwalla, Feroze; Venkatraman, Srikanth; Edmondson, Scott D

Design and Synthesis of Novel, Selective GPR40 AgoPAMs

新型选择性GPR40 AgoPAMs的设计与合成

Plummer, Christopher W; Clements, Matthew J; Chen, Helen; Rajagopalan, Murali; Josien, Hubert; Hagmann, William K; Miller, Michael; Trujillo, Maria E; Kirkland, Melissa; Kosinski, Daniel; Mane, Joel; Pachanski, Michele; Cheewatrakoolpong, Boonlert; Nolting, Andrew F; Orr, Robert; Christensen, Melodie; Campeau, Louis-Charles; Wright, Michael J; Bugianesi, Randal; Souza, Sarah; Zhang, Xiaoping; Di Salvo, Jerry; Weinglass, Adam B; Tschirret-Guth, Richard; Nargund, Ravi; Howard, Andrew D; Colletti, Steven L

GPR40 partial agonist MK-2305 lower fasting glucose in the Goto Kakizaki rat via suppression of endogenous glucose production

GPR40 部分激动剂 MK-2305 通过抑制内源性葡萄糖生成降低 Goto Kakizaki 大鼠的空腹血糖

Corin Miller, Michele J Pachanski, Melissa E Kirkland, Daniel T Kosinski, Joel Mane, Michelle Bunzel, Jin Cao, Sarah Souza, Brande Thomas-Fowlkes, Jerry Di Salvo, Adam B Weinglass, Xiaoyan Li, Robert W Myers, Kevin Knagge, Paul E Carrington, William K Hagmann, Maria E Trujillo

GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent

GPR40 部分激动剂和 AgoPAM:对啮齿动物葡萄糖和激素分泌的不同影响

Michele J Pachanski, Melissa E Kirkland, Daniel T Kosinski, Joel Mane, Boonlert Cheewatrakoolpong, Jiyan Xue, Daphne Szeto, Gail Forrest, Corin Miller, Michelle Bunzel, Christopher W Plummer, Harry R Chobanian, Michael W Miller, Sarah Souza, Brande S Thomas-Fowlkes, Aimie M Ogawa, Adam B Weinglass,