日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fragment-Based Approach to Targeting Inosine-5'-monophosphate Dehydrogenase (IMPDH) from Mycobacterium tuberculosis

基于片段的方法靶向结核分枝杆菌的肌苷-5'-单磷酸脱氢酶(IMPDH)

Trapero, Ana; Pacitto, Angela; Singh, Vinayak; Sabbah, Mohamad; Coyne, Anthony G; Mizrahi, Valerie; Blundell, Tom L; Ascher, David B; Abell, Chris

The Inosine Monophosphate Dehydrogenase, GuaB2, Is a Vulnerable New Bactericidal Drug Target for Tuberculosis

肌苷单磷酸脱氢酶 GuaB2 是结核病新型杀菌药物的易损靶点

Singh, Vinayak; Donini, Stefano; Pacitto, Angela; Sala, Claudia; Hartkoorn, Ruben C; Dhar, Neeraj; Keri, Gyorgy; Ascher, David B; Mondésert, Guillaume; Vocat, Anthony; Lupien, Andréanne; Sommer, Raphael; Vermet, Hélène; Lagrange, Sophie; Buechler, Joe; Warner, Digby F; McKinney, John D; Pato, Janos; Cole, Stewart T; Blundell, Tom L; Rizzi, Menico; Mizrahi, Valerie

Lst4, the yeast Fnip1/2 orthologue, is a DENN-family protein.

Lst4 是酵母 Fnip1/2 的直系同源物,属于 DENN 家族蛋白

Pacitto Angela, Ascher David B, Wong Louise H, Blaszczyk Beata K, Nookala Ravi K, Zhang Nianshu, Dokudovskaya Svetlana, Levine Tim P, Blundell Tom L

Crystal structure of folliculin reveals a hidDENN function in genetically inherited renal cancer

卵泡蛋白的晶体结构揭示了其在遗传性肾癌中的隐藏功能

Nookala, Ravi K; Langemeyer, Lars; Pacitto, Angela; Ochoa-Montaño, Bernardo; Donaldson, Jane C; Blaszczyk, Beata K; Chirgadze, Dimitri Y; Barr, Francis A; Bazan, J Fernando; Blundell, Tom L