日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Comparative pharmacokinetics and pharmacodynamics of intravenous artelinate versus artesunate in uncomplicated Plasmodium coatneyi-infected rhesus monkey model

在无并发症的科氏疟原虫感染的恒河猴模型中,静脉注射阿替林与青蒿琥酯的药代动力学和药效学比较

Teja-Isavadharm, Paktiya; Siriyanonda, Duangsuda; Rasameesoraj, Maneerat; Limsalakpeth, Amporn; Chanarat, Nitima; Komcharoen, Natthasorn; Weina, Peter J; Saunders, David L; Gettayacamin, Montip; Scott Miller, R

Ex Vivo Drug Susceptibility Testing and Molecular Profiling of Clinical Plasmodium falciparum Isolates from Cambodia from 2008 to 2013 Suggest Emerging Piperaquine Resistance

2008年至2013年间柬埔寨临床分离的恶性疟原虫的体外药物敏感性试验和分子谱分析表明,哌喹耐药性正在出现。

Chaorattanakawee, Suwanna; Saunders, David L; Sea, Darapiseth; Chanarat, Nitima; Yingyuen, Kritsanai; Sundrakes, Siratchana; Saingam, Piyaporn; Buathong, Nillawan; Sriwichai, Sabaithip; Chann, Soklyda; Se, Youry; Yom, You; Heng, Thay Kheng; Kong, Nareth; Kuntawunginn, Worachet; Tangthongchaiwiriya, Kuntida; Jacob, Christopher; Takala-Harrison, Shannon; Plowe, Christopher; Lin, Jessica T; Chuor, Char Meng; Prom, Satharath; Tyner, Stuart D; Gosi, Panita; Teja-Isavadharm, Paktiya; Lon, Chanthap; Lanteri, Charlotte A

Randomized, double-blind, placebo-controlled clinical trial of a two-day regimen of dihydroartemisinin-piperaquine for malaria prevention halted for concern over prolonged corrected QT interval

一项为期两天的双氢青蒿素-哌喹方案预防疟疾的随机、双盲、安慰剂对照临床试验,因担心校正QT间期延长而中止。

Manning, Jessica; Vanachayangkul, Pattaraporn; Lon, Chanthap; Spring, Michele; So, Mary; Sea, Darapiseth; Se, Youry; Somethy, Sok; Phann, Sut-Thang; Chann, Soklyda; Sriwichai, Sabaithip; Buathong, Nillawan; Kuntawunginn, Worachet; Mitprasat, Mashamon; Siripokasupkul, Raveewan; Teja-Isavadharm, Paktiya; Soh, Eugene; Timmermans, Ans; Lanteri, Charlotte; Kaewkungwal, Jaranit; Auayporn, Montida; Tang, Douglas; Chour, Char Meng; Prom, Satharath; Haigney, Mark; Cantilena, Louis; Saunders, David

Pharmacokinetics and pharmacodynamics of (+)-primaquine and (-)-primaquine enantiomers in rhesus macaques (Macaca mulatta)

恒河猴(Macaca mulatta)体内(+)-伯氨喹和(-)-伯氨喹对映异构体的药代动力学和药效学研究

Saunders, David; Vanachayangkul, Pattaraporn; Imerbsin, Rawiwan; Khemawoot, Phisit; Siripokasupkul, Raveewan; Tekwani, Babu L; Sampath, Aruna; Nanayakkara, N P Dhammika; Ohrt, Colin; Lanteri, Charlotte; Gettyacamin, Montip; Teja-Isavadharm, Paktiya; Walker, Larry

Pharmacokinetic evaluation of intravenous artesunate in adults with uncomplicated falciparum malaria in Kenya: a phase II study

肯尼亚成人单纯性恶性疟疾患者静脉注射青蒿琥酯的药代动力学评价:一项II期研究

Li, Qigui; Remich, Shon; Miller, Scott R; Ogutu, Bernhards; Otieno, Walter; Melendez, Victor; Teja-Isavadharm, Paktiya; Weina, Peter J; Hickman, Mark R; Smith, Bryan; Polhemus, Mark

Anti-relapse activity of mirincamycin in the Plasmodium cynomolgi sporozoite-infected Rhesus monkey model

米林霉素在感染猕猴疟原虫子孢子的恒河猴模型中的抗复发活性

Fracisco, Susan; Teja-isavadharm, Paktiya; Gettayacamin, Montip; Berman, Jonathan; Li, Qigui; Melendez, Victor; Saunders, David; Xie, Lisa; Ohrt, Colin

Pharmacokinetics and pharmacodynamics of oral artesunate monotherapy in patients with uncomplicated Plasmodium falciparum malaria in western Cambodia

柬埔寨西部地区单纯性恶性疟疾患者口服青蒿琥酯单药治疗的药代动力学和药效学研究

Saunders, David; Khemawoot, Phisit; Vanachayangkul, Pattaraporn; Siripokasupkul, Raveewan; Bethell, Delia; Tyner, Stuart; Se, Youry; Rutvisuttinunt, Wiriya; Sriwichai, Sabaithip; Chanthap, Lon; Lin, Jessica; Timmermans, Ans; Socheat, Doung; Ringwald, Pascal; Noedl, Harald; Smith, Bryan; Fukuda, Mark; Teja-Isavadharm, Paktiya

Optimizing the HRP-2 in vitro malaria drug susceptibility assay using a reference clone to improve comparisons of Plasmodium falciparum field isolates

利用参考克隆优化HRP-2体外疟疾药物敏感性试验,以改进恶性疟原虫野外分离株的比较。

Rutvisuttinunt, Wiriya; Chaorattanakawee, Suwanna; Tyner, Stuart D; Teja-Isavadharm, Paktiya; Se, Youry; Yingyuen, Kritsanai; Chaichana, Panjaporn; Bethell, Delia; Walsh, Douglas S; Lon, Chanthap; Fukuda, Mark; Socheat, Duong; Noedl, Harald; Schaecher, Kurt; Saunders, David L