Structure-Based Design of CBP/EP300 Degraders: When Cooperativity Overcomes Affinity
基于结构的CBP/EP300降解剂设计:当协同性战胜亲和性
期刊:JACS Au
影响因子:8.7
doi:10.1021/jacsau.4c00292
Cheng-Sánchez, Iván; Gosselé, Katherine; Palaferri, Leonardo; Laul, Eleen; Riccabella, Gionata; Bedi, Rajiv K; Li, Yaozong; Müller, Anna; Corbeski, Ivan; Caflisch, Amedeo; Nevado, Cristina