日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Evaluation of ASC as a therapeutic target for Alzheimer's disease

评估ASC作为阿尔茨海默病治疗靶点的潜力

Clayton, W Brent; Kulas, Joshua A; Liu, Jiahui; Walia, Nidhi; Rangel-Barajas, Claudia; Johnson, Travis; Zhang, Jie; Huang, Kun; Mesecar, Andrew D; Dage, Jeffrey L; Lamb, Bruce T; Palkowitz, Alan D; Richardson, Timothy I

Next-generation Alzheimer's therapeutics: target assessment and enablement at the Indiana University School of Medicine-Purdue University TREAT-AD Center

下一代阿尔茨海默病疗法:印第安纳大学医学院-普渡大学TREAT-AD中心的靶点评估和开发

Richardson, Timothy I; Klein, Rebecca C; Huang, Kun; Zhang, Jie; Mesecar, Andrew D; Dage, Jeffrey L; Clayton, Brent; Lamb, Bruce T; Palkowitz, Alan D

From consortia discovery to biotech creation: An innovative approach to next-gen Alzheimer's drugs

从联盟发现到生物技术创造:下一代阿尔茨海默病药物的创新方法

Giardina, Sarah F; Culver, Alexander; Ahmed, Chandrama; Mirescu, Christian; Oblak, Adrian L; Brosch, Jared; Clayton, W Brent; Dage, Jeffrey L; Lamb, Bruce T; Richardson, Timothy I; Small, Derek; Palkowitz, Alan D

Generation and characterization of iPSC-derived microglia for in vitro modeling of stimuli-specific neuroimmune responses.

利用 iPSC 衍生的小胶质细胞进行体外模型构建,以模拟刺激特异性神经免疫反应。

Haskell Angela K, Kulas Joshua A, Carter William E, Javens-Wolfe June, Hinkel Raven Dance, Moussaif Mustapha, Smiley Jacob S, Lazaro Olivia, Robertson Sylvia, Palkowitz Alan D, Lamb Bruce T, Richardson Timothy I, Dage Jeffrey L, Chu Shaoyou, Johnson Travis, Stancato Louis F, Syed Abdul Qadir

Optimization and Characterization of SHIP1 Ligands for Cellular Target Engagement and Activity in Alzheimer's Disease Models.

SHIP1 配体的优化和表征及其在阿尔茨海默病模型中的细胞靶点结合和活性。

Jesudason Cynthia D, Rangel-Barajas Claudia, Beach Colin J, Beck Daniel E, Caballero-Floran Isaac H, Clayton W Brent, Da Silva Lais, David Juliane C, Doolen Suzanne, Faulkner Alexandra N, Hamdani Adam K, Huhe Hasi, Huynh Kevin, Imhoff Ryan D, Javens-Wolfe June, Mason Emily R, Moussaif Mustapha, Singhal Kratika, Soni Disha M, van Buuren-Milne Matilda, Williams Sean-Paul, Angus Steven P, Chu Shaoyou, Dage Jeffrey L, Hipskind Philip A, Johnson Travis S, Kaddurah-Daouk Rima, Lamb Bruce T, Meikle Peter J, Mesecar Andrew D, Palkowitz Alan D, Quinney Sara K, Sukoff Rizzo Stacey J, Oblak Adrian L, Richardson Timothy I

Accelerating Medicinal Chemistry: A C(sp(3))-Rich Fragment Toolbox for Redox-Neutral Cross-Coupling

加速药物化学:富含 AC(sp(3)) 的片段工具箱用于氧化还原中性交叉偶联

Tsien, Jet; Péter, Áron; Zeng, Xin; Wang, Shuanghu; Jiang, Baiyang; Emmanuel, Megan A; Oderinde, Martins S; Bolduc, Philippe N; Nicastri, Michael C; Dey, Shalini; Collins, Michael R; Lee, Johnny W; Bravo, Martin; Richardson, Paul F; Sach, Neal W; Bernier, Louise; Palkowitz, Maximilian D; Qiao, Jennifer X; Kawamata, Yu; Baran, Phil S

Diversity-Oriented C-H Activation Reactions of the Naphthalene Scaffold

萘骨架的多样性导向CH活化反应

Fan, Zhoulong; Hoque, Md Emdadul; Wu, Kevin; Palkowitz, Maximilian D; Velaparthi, Upender; Gillman, Kevin W; Qiao, Jennifer X; Yu, Jin-Quan

Identification of PLCγ2 activators for the treatment of Alzheimer’s disease

鉴定用于治疗阿尔茨海默病的PLCγ2激活剂

Hawksley, J C; Clayton, Brent; Massey, Steven M; Chu, Shaoyou; Mason, Emily R; Bissel, Stephanie J; Bedford, Logan M; Rizzo, Stacey J Sukoff; Mesecar, Andrew D; Kaiser, Bridget L; Lendy, Emma K; Lamb, Bruce T; Palkowitz, Alan D; Richardson, Timothy I

Discovery of N-X anomeric amides as electrophilic halogenation reagents

发现NX异头酰胺作为亲电卤化试剂

Wang, Yu; Bi, Cheng; Kawamata, Yu; Grant, Lauren N; Samp, Lacey; Richardson, Paul F; Zhang, Shasha; Harper, Kaid C; Palkowitz, Maximilian D; Vasilopoulos, Aristidis; Collins, Michael R; Oderinde, Martins S; Tyrol, Chet C; Chen, Doris; LaChapelle, Erik A; Bailey, Jake B; Qiao, Jennifer X; Baran, Phil S

In vitro plaque formation model to unravel biofilm formation dynamics on implant abutment surfaces

体外菌斑形成模型揭示种植体基台表面生物膜形成的动态过程

Utomo, Romualdus Nugraha Catur; Palkowitz, Alena Lisa; Gan, Lin; Rudzinski, Anna; Franzen, Julia; Ballerstedt, Hendrik; Zimmermann, Martin; Blank, Lars Mathias; Fischer, Horst; Wolfart, Stefan; Tuna, Taskin