日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Reversible male contraception by targeted inhibition of serine/threonine kinase 33

通过靶向抑制丝氨酸/苏氨酸激酶33实现可逆性男性避孕

Ku, Angela F; Sharma, Kiran L; Ta, Hai Minh; Sutton, Courtney M; Bohren, Kurt M; Wang, Yong; Chamakuri, Srinivas; Chen, Ruihong; Hakenjos, John M; Jimmidi, Ravikumar; Kent, Katarzyna; Li, Feng; Li, Jian-Yuan; Ma, Lang; Madasu, Chandrashekhar; Palaniappan, Murugesan; Palmer, Stephen S; Qin, Xuan; Robers, Matthew B; Sankaran, Banumathi; Tan, Zhi; Vasquez, Yasmin M; Wang, Jian; Wilkinson, Jennifer; Yu, Zhifeng; Ye, Qiuji; Young, Damian W; Teng, Mingxing; Kim, Choel; Matzuk, Martin M

Discovery of highly potent and ALK2/ALK1 selective kinase inhibitors using DNA-encoded chemistry technology.

利用DNA编码化学技术发现高效且对ALK2/ALK1具有选择性的激酶抑制剂

Jimmidi Ravikumar, Monsivais Diana, Ta Hai Minh, Sharma Kiran L, Bohren Kurt M, Chamakuri Srinivas, Liao Zian, Li Feng, Hakenjos John M, Li Jian-Yuan, Mishina Yuji, Pan Haichun, Qin Xuan, Robers Matthew B, Sankaran Banumathi, Tan Zhi, Tang Suni, Vasquez Yasmin M, Wilkinson Jennifer, Young Damian W, Palmer Stephen S, MacKenzie Kevin R, Kim Choel, Matzuk Martin M

Discovery of potent BET bromodomain 1 stereoselective inhibitors using DNA-encoded chemical library selections

利用DNA编码化学库筛选发现强效BET溴结构域1立体选择性抑制剂

Modukuri, Ram K; Yu, Zhifeng; Tan, Zhi; Ta, Hai Minh; Ucisik, Melek Nihan; Jin, Zhuang; Anglin, Justin L; Sharma, Kiran L; Nyshadham, Pranavanand; Li, Feng; Riehle, Kevin; Faver, John C; Duong, Kevin; Nagarajan, Sureshbabu; Simmons, Nicholas; Palmer, Stephen S; Teng, Mingxing; Young, Damian W; Yi, Joanna S; Kim, Choel; Matzuk, Martin M

Discovery and characterization of bromodomain 2-specific inhibitors of BRDT

BRDT溴结构域2特异性抑制剂的发现与表征

Yu, Zhifeng; Ku, Angela F; Anglin, Justin L; Sharma, Rajesh; Ucisik, Melek Nihan; Faver, John C; Li, Feng; Nyshadham, Pranavanand; Simmons, Nicholas; Sharma, Kiran L; Nagarajan, Sureshbabu; Riehle, Kevin; Kaur, Gundeep; Sankaran, Banumathi; Storl-Desmond, Marta; Palmer, Stephen S; Young, Damian W; Kim, Choel; Matzuk, Martin M

DNA-encoded chemistry technology yields expedient access to SARS-CoV-2 M(pro) inhibitors.

DNA编码化学技术可快速获得SARS-CoV-2 M(pro)抑制剂

Chamakuri Srinivas, Lu Shuo, Ucisik Melek Nihan, Bohren Kurt M, Chen Ying-Chu, Du Huang-Chi, Faver John C, Jimmidi Ravikumar, Li Feng, Li Jian-Yuan, Nyshadham Pranavanand, Palmer Stephen S, Pollet Jeroen, Qin Xuan, Ronca Shannon E, Sankaran Banumathi, Sharma Kiran L, Tan Zhi, Versteeg Leroy, Yu Zhifeng, Matzuk Martin M, Palzkill Timothy, Young Damian W

Follicle-Stimulating Hormone Induces Lipid Droplets via Gαi/o and β-Arrestin in an Endometrial Cancer Cell Line

促卵泡激素通过 Gαi/o 和 β-arrestin 诱导子宫内膜癌细胞系中脂滴的形成

Sayers, Niamh S; Anujan, Priyanka; Yu, Henry N; Palmer, Stephen S; Nautiyal, Jaya; Franks, Stephen; Hanyaloglu, Aylin C

Bentamapimod (JNK Inhibitor AS602801) Induces Regression of Endometriotic Lesions in Animal Models

Bentamapimod(JNK抑制剂AS602801)可诱导动物模型中子宫内膜异位症病灶消退

Palmer, Stephen S; Altan, Melis; Denis, Deborah; Tos, Enrico Gillio; Gotteland, Jean-Pierre; Osteen, Kevin G; Bruner-Tran, Kaylon L; Nataraja, Selvaraj G

Discovery and Development of Small Molecule Allosteric Modulators of Glycoprotein Hormone Receptors

糖蛋白激素受体小分子变构调节剂的发现与开发

Nataraja, Selvaraj G; Yu, Henry N; Palmer, Stephen S

Biomarkers in reproductive medicine: the promise, and can it be fulfilled?

生殖医学中的生物标志物:前景如何?能否实现?

Palmer, Stephen S; Barnhart, Kurt T

Follicle-stimulating hormone activates extracellular signal-regulated kinase but not extracellular signal-regulated kinase kinase through a 100-kDa phosphotyrosine phosphatase

卵泡刺激素通过一种100 kDa的磷酸酪氨酸磷酸酶激活细胞外信号调节激酶(ERK),但不激活细胞外信号调节激酶激酶(ERKK)。

Cottom, Joshua; Salvador, Lisa M; Maizels, Evelyn T; Reierstad, Scott; Park, Youngkyu; Carr, Daniel W; Davare, Monika A; Hell, Johannes W; Palmer, Stephen S; Dent, Paul; Kawakatsu, Hisaaki; Ogata, Masato; Hunzicker-Dunn, Mary