日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Polymer Systems with Correlated Activity: Stars Versus Linear Chains

具有相关活性的聚合物体系:星形聚合物与线性链聚合物

Buglakov, Aleksandr I; Chuphal, Prabha; Rudyak, Vladimir Yu; Chertovich, Alexander V; Palyulin, Vladimir V

Conjugates of amiridine and salicylic derivatives as promising multifunctional CNS agents for potential treatment of Alzheimer's disease.

脒基脒和水杨酸衍生物的结合物作为有前景的多功能中枢神经系统药物,可用于治疗阿尔茨海默病

Makhaeva Galina F, Grishchenko Maria V, Kovaleva Nadezhda V, Boltneva Natalia P, Rudakova Elena V, Astakhova Tatiana Y, Timokhina Elena N, Pronkin Pavel G, Lushchekina Sofya V, Khudina Olga G, Zhilina Ekaterina F, Shchegolkov Evgeny V, Lapshina Maria A, Dubrovskaya Elena S, Radchenko Eugene V, Palyulin Vladimir A, Burgart Yanina V, Saloutin Victor I, Charushin Valery N, Richardson Rudy J

Free Energy Barriers for Passive Drug Transport through the Mycobacterium tuberculosis Outer Membrane: A Molecular Dynamics Study

结核分枝杆菌外膜被动药物转运的自由能垒:分子动力学研究

Steshin, Ilya S; Vasyankin, Alexander V; Shirokova, Ekaterina A; Rozhkov, Alexey V; Livshits, Grigory D; Panteleev, Sergey V; Radchenko, Eugene V; Ignatov, Stanislav K; Palyulin, Vladimir A

Temperature-Induced Restructuring of Mycolic Acid Bilayers Modeling the Mycobacterium tuberculosis Outer Membrane: A Molecular Dynamics Study

温度诱导的模拟结核分枝杆菌外膜的分枝菌酸双层结构重构:分子动力学研究

Vasyankin, Alexander V; Panteleev, Sergey V; Steshin, Ilya S; Shirokova, Ekaterina A; Rozhkov, Alexey V; Livshits, Grigory D; Radchenko, Eugene V; Ignatov, Stanislav K; Palyulin, Vladimir A

Features of DNA-Montmorillonite Binding Visualized by Atomic Force Microscopy

利用原子力显微镜观察DNA-蒙脱石结合的特征

Kraevsky, Sergey V; Barinov, Nikolay A; Morozova, Olga V; Palyulin, Vladimir V; Kremleva, Alena V; Klinov, Dmitry V

5-Nitroisoxazoles in S(N)Ar Reactions: A Novel Chemo- and Regioselective Approach to Isoxazole-Based Bivalent Ligands of AMPA Receptors

5-硝基异噁唑在S(N)Ar反应中的应用:一种新型的基于异噁唑的AMPA受体二价配体的化学选择性和区域选择性合成方法

Vasilenko, Dmitry A; Temnyakova, Nadezhda S; Dronov, Sevastian E; Radchenko, Eugene V; Grishin, Yuri K; Gabrel'yan, Alexey V; Zamoyski, Vladimir L; Grigoriev, Vladimir V; Averina, Elena B; Palyulin, Vladimir A

Derivatives of 9-phosphorylated acridine as butyrylcholinesterase inhibitors with antioxidant activity and the ability to inhibit β-amyloid self-aggregation: potential therapeutic agents for Alzheimer's disease

9-磷酸化吖啶衍生物作为丁酰胆碱酯酶抑制剂,具有抗氧化活性并能抑制β-淀粉样蛋白自聚集:阿尔茨海默病潜在的治疗药物

Makhaeva, Galina F; Kovaleva, Nadezhda V; Rudakova, Elena V; Boltneva, Natalia P; Lushchekina, Sofya V; Astakhova, Tatiana Yu; Timokhina, Elena N; Serebryakova, Olga G; Shchepochkin, Alexander V; Averkov, Maxim A; Utepova, Irina A; Demina, Nadezhda S; Radchenko, Eugene V; Palyulin, Vladimir A; Fisenko, Vladimir P; Bachurin, Sergey O; Chupakhin, Oleg N; Charushin, Valery N; Richardson, Rudy J

Conformational Dynamics and Stability of Bilayers Formed by Mycolic Acids from the Mycobacterium tuberculosis Outer Membrane

结核分枝杆菌外膜分枝菌酸形成的双层膜的构象动力学和稳定性

Savintseva, Liana A; Steshin, Ilya S; Avdoshin, Alexander A; Panteleev, Sergey V; Rozhkov, Alexey V; Shirokova, Ekaterina A; Livshits, Grigory D; Vasyankin, Alexander V; Radchenko, Eugene V; Ignatov, Stanislav K; Palyulin, Vladimir A

New Allosteric Modulators of AMPA Receptors: Synthesis and Study of Their Functional Activity by Radioligand-Receptor Binding Analysis

AMPA 受体的新型变构调节剂:合成并通过放射性配体-受体结合分析研究其功能活性

Elena A Golubeva, Mstislav I Lavrov, Polina N Veremeeva, Tatiana V Vyunova, Konstantin V Shevchenko, Maxim A Topchiy, Andrey F Asachenko, Vladimir A Palyulin

Conjugates of Tacrine and Salicylic Acid Derivatives as New Promising Multitarget Agents for Alzheimer's Disease

他克林与水杨酸衍生物的结合物作为治疗阿尔茨海默病的新型有前途的多靶点药物

Galina F Makhaeva, Nadezhda V Kovaleva, Elena V Rudakova, Natalia P Boltneva, Maria V Grishchenko, Sofya V Lushchekina, Tatiana Y Astakhova, Olga G Serebryakova, Elena N Timokhina, Ekaterina F Zhilina, Evgeny V Shchegolkov, Mariya V Ulitko, Eugene V Radchenko, Vladimir A Palyulin, Yanina V Burgart,