日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Pharmacology of a Morphinan-Derived Dual Mu-Kappa Opioid Receptor Agonist Analgesic.

吗啡烷衍生的双重μ-κ阿片受体激动剂镇痛药的合成与药理学研究

Varga Balazs R, Uprety Rajendra, Paul Barnali, Knoll Alexis, Ramos-Gonzalez Nokomis, Appourchaux Kevin, Taylor Tori, Turgutalp Bengisu, Shinouchi Ryosuke, Eans Shainnel O, Williams Ashai K, Vasquez-Grinnell Steven G, Zaidi Saheem, Nazarova Antonina L, Varadi Andras, Le Rouzic Valerie, Brown Taylor G, Martinez Shani, Ansonoff Michael, Dardashti Rebecca Notis, Hunkele Amanda, Subrath Joan, Welch Matthew, Xu Jin, Rossi Grace C, Pintar John, Pasternak Gavril W, Katritch Vsevolod, McLaughlin Jay P, Pan Ying Xian, Majumdar Susruta

Elevating levels of the endocannabinoid 2-arachidonoylglycerol blunts opioid reward but not analgesia

提高内源性大麻素 2-花生四烯酸甘油酯的水平会减弱阿片类药物的奖赏效应,但不会减弱其镇痛作用。

Martínez-Rivera, Arlene; Fetcho, Robert N; Birmingham, Lizzie; Xu, Jin; Yang, Ruirong; Foord, Careen; Scala-Chávez, Diego; Mekawy, Narmin; Pleil, Kristen; Pickel, Virginia M; Liston, Conor; Castorena, Carlos M; Levitz, Joshua; Pan, Ying-Xian; Briand, Lisa A; Rajadhyaksha, Anjali M; Lee, Francis S

Photo-affinity and Metabolic Labeling Probes Based on the Opioid Alkaloids

基于阿片生物碱的光亲和和代谢标记探针

Duque, Mark Anthony Leon; Vallavoju, Nandini; Zhang, Tiffany; Yvon, Robert; Pan, Ying-Xian; Woo, Christina M

Structure-based design of bitopic ligands for the µ-opioid receptor

基于结构的μ-阿片受体双位点配体设计

Faouzi, Abdelfattah; Wang, Haoqing; Zaidi, Saheem A; DiBerto, Jeffrey F; Che, Tao; Qu, Qianhui; Robertson, Michael J; Madasu, Manish K; El Daibani, Amal; Varga, Balazs R; Zhang, Tiffany; Ruiz, Claudia; Liu, Shan; Xu, Jin; Appourchaux, Kevin; Slocum, Samuel T; Eans, Shainnel O; Cameron, Michael D; Al-Hasani, Ream; Pan, Ying Xian; Roth, Bryan L; McLaughlin, Jay P; Skiniotis, Georgios; Katritch, Vsevolod; Kobilka, Brian K; Majumdar, Susruta

Binding preference at the μ-opioid receptor underlies distinct pharmacology of cyclopropyl versus valeryl analogs of fentanyl

芬太尼环丙基类似物与戊酰基类似物在μ-阿片受体上的结合偏好是其药理学差异的根本原因。

Xie, Bing; Le Rouzic, Valerie P; Goldberg, Alexander; Tsai, Meng-Hua M; Chen, Li; Zhang, Tiffany; Sinha, Antara; Pan, Ying-Xian; Baumann, Michael H; Shi, Lei

Exploring Pharmacological Functions of Alternatively Spliced Variants of the Mu Opioid Receptor Gene, Oprm1, via Gene-Targeted Animal Models

利用基因靶向动物模型探索μ阿片受体基因Oprm1选择性剪接变体的药理功能

Kang, Wenjian; Liu, Shan; Xu, Jin; Abrimian, Anna; Malik, Ayma F; Chien, Raymond; Adaralegbe, Adejuyigbe; Amponsah, Akwasi; Cartegni, Luca; Pintar, John; Pan, Ying-Xian

Dysregulated expression of the alternatively spliced variant mRNAs of the mu opioid receptor gene, OPRM1, in the medial prefrontal cortex of male human heroin abusers and heroin self-administering male rats

男性海洛因滥用者和海洛因自我给药雄性大鼠内侧前额皮质中μ阿片受体基因OPRM1选择性剪接变体mRNA的表达失调

Brown, Taylor G; Xu, Jin; Hurd, Yasmin L; Pan, Ying-Xian

From Pharmacology to Physiology: Endocrine Functions of μ-Opioid Receptor Networks

从药理学到生理学:μ-阿片受体网络的内分泌功能

Jaschke, Nikolai; Pählig, Sophie; Pan, Ying-Xian; Hofbauer, Lorenz C; Göbel, Andy; Rachner, Tilman D

Endogenous Opioid Peptides and Alternatively Spliced Mu Opioid Receptor Seven Transmembrane Carboxyl-Terminal Variants

内源性阿片肽和选择性剪接的μ阿片受体七次跨膜羧基末端变体

Abrimian, Anna; Kraft, Tamar; Pan, Ying-Xian

Alternative Pre-mRNA Splicing of the Mu Opioid Receptor Gene, OPRM1: Insight into Complex Mu Opioid Actions

μ阿片受体基因OPRM1的mRNA选择性剪接:深入了解复杂的μ阿片受体作用

Liu, Shan; Kang, Wen-Jia; Abrimian, Anna; Xu, Jin; Cartegni, Luca; Majumdar, Susruta; Hesketh, Patrick; Bekker, Alex; Pan, Ying-Xian