日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate

三氨基嘧啶是一种速效且长效的抗疟疾候选药物。

Hameed P, Shahul; Solapure, Suresh; Patil, Vikas; Henrich, Philipp P; Magistrado, Pamela A; Bharath, Sowmya; Murugan, Kannan; Viswanath, Pavithra; Puttur, Jayashree; Srivastava, Abhishek; Bellale, Eknath; Panduga, Vijender; Shanbag, Gajanan; Awasthy, Disha; Landge, Sudhir; Morayya, Sapna; Koushik, Krishna; Saralaya, Ramanatha; Raichurkar, Anandkumar; Rautela, Nikhil; Roy Choudhury, Nilanjana; Ambady, Anisha; Nandishaiah, Radha; Reddy, Jitendar; Prabhakar, K R; Menasinakai, Sreenivasaiah; Rudrapatna, Suresh; Chatterji, Monalisa; Jiménez-Díaz, María Belén; Martínez, María Santos; Sanz, Laura María; Coburn-Flynn, Olivia; Fidock, David A; Lukens, Amanda K; Wirth, Dyann F; Bandodkar, Balachandra; Mukherjee, Kakoli; McLaughlin, Robert E; Waterson, David; Rosenbrier-Ribeiro, Lyn; Hickling, Kevin; Balasubramanian, V; Warner, Peter; Hosagrahara, Vinayak; Dudley, Adam; Iyer, Pravin S; Narayanan, Shridhar; Kavanagh, Stefan; Sambandamurthy, Vasan K

In silico-based high-throughput screen for discovery of novel combinations for tuberculosis treatment

利用计算机模拟高通量筛选发现治疗结核病的新组合

Singh, Ragini; Ramachandran, Vasanthi; Shandil, Radha; Sharma, Sreevalli; Khandelwal, Swati; Karmarkar, Malancha; Kumar, Naveen; Solapure, Suresh; Saralaya, Ramanatha; Nanduri, Robert; Panduga, Vijender; Reddy, Jitendar; Prabhakar, K R; Rajagopalan, Swaminathan; Rao, Narasimha; Narayanan, Shridhar; Anandkumar, Anand; Balasubramanian, V; Datta, Santanu

MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants

MK-5172,一种选择性抑制丙型肝炎病毒NS3/4a蛋白酶的药物,对多种基因型和耐药变异株均具有广泛活性。

Draper, Michael P; Weir, S; Macone, A; Donatelli, J; Trieber, C A; Tanaka, S K; Levy, Stuart B; P, Shahul Hameed; Solapure, Suresh; Mukherjee, Kakoli; Nandi, Vrinda; Waterson, David; Shandil, Radha; Balganesh, Meenakshi; Sambandamurthy, Vasan K; Raichurkar, Anand Kumar; Deshpande, Abhijeet; Ghosh, Anirban; Awasthy, Disha; Shanbhag, Gajanan; Sheikh, Gulebahar; McMiken, Helen; Puttur, Jayashree; Reddy, Jitendar; Werngren, Jim; Read, Jon; Kumar, Mahesh; R, Manjunatha; Chinnapattu, Murugan; Madhavapeddi, Prashanti; Manjrekar, Praveena; Basu, Reetobrata; Gaonkar, Sheshagiri; Sharma, Sreevalli; Hoffner, Sven; Humnabadkar, Vaishali; Subbulakshmi, Venkita; Panduga, Vijender; Summa, Vincenzo; Ludmerer, Steven W; McCauley, John A; Fandozzi, Christine; Burlein, Christine; Claudio, Giuliano; Coleman, Paul J; DiMuzio, Jillian M; Ferrara, Marco; Filippo, Marcello Di; Gates, Adam T; Graham, Donald J; Harper, Steven; Hazuda, Daria J; Huang, Qian; McHale, Carolyn; Monteagudo, Edith; Pucci, Vincenzo; Rowley, Michael; Rudd, Michael T; Soriano, Aileen; Stahlhut, Mark W; Vacca, Joseph P; Olsen, David B; Liverton, Nigel J; Carroll, Steven S

1,4-azaindole, a potential drug candidate for treatment of tuberculosis

1,4-氮杂吲哚,一种潜在的结核病治疗候选药物

Chatterji, Monalisa; Shandil, Radha; Manjunatha, M R; Solapure, Suresh; Ramachandran, Vasanthi; Kumar, Naveen; Saralaya, Ramanatha; Panduga, Vijender; Reddy, Jitendar; Prabhakar, K R; Sharma, Sreevalli; Sadler, Claire; Cooper, Christopher B; Mdluli, Khisi; Iyer, Pravin S; Narayanan, Shridhar; Shirude, Pravin S

In vitro and in vivo efficacy of β-lactams against replicating and slowly growing/nonreplicating Mycobacterium tuberculosis

β-内酰胺类抗生素对复制型和生长缓慢/非复制型结核分枝杆菌的体外和体内疗效

Solapure, Suresh; Dinesh, Neela; Shandil, Radha; Ramachandran, Vasanthi; Sharma, Sreevalli; Bhattacharjee, Deepa; Ganguly, Samit; Reddy, Jitendar; Ahuja, Vijaykamal; Panduga, Vijender; Parab, Manish; Vishwas, K G; Kumar, Naveen; Balganesh, Meenakshi; Balasubramanian, V

Effect of coadministration of moxifloxacin and rifampin on Mycobacterium tuberculosis in a murine aerosol infection model

莫西沙星和利福平联合用药对小鼠气溶胶感染模型中结核分枝杆菌的影响

Balasubramanian, V; Solapure, S; Gaonkar, S; Mahesh Kumar, K N; Shandil, R K; Deshpande, Abhijeet; Kumar, Naveen; Vishwas, K G; Panduga, Vijender; Reddy, Jitendar; Ganguly, Samit; Louie, A; Drusano, G L