Addressing the Intracellular Vestibule of the Plasmodial Lactate Transporter PfFNT by p-Substituted Inhibitors Amplifies In Vitro Activity
通过对质粒乳酸转运蛋白 PfFNT 的细胞内前庭进行 p-取代抑制剂处理,可增强其体外活性。
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c01674
Nerlich, Cornelius; Tiedjens, Finn; Hertel, Robin; Henke, Björn; Häuer, Susan; Panitzsch, Lea S; Hansen, Kerrin; Franck, Ole; Mete, Antonio; Leroy, Didier; Schade, Dennis; Peifer, Christian; Hannus, Stefan; Becker, Frank; Wittlin, Sergio; Spielmann, Tobias; Beitz, Eric