日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An allosteric inhibitor of the Zika virus NS2B-NS3 protease with oral efficacy in mouse models

一种寨卡病毒NS2B-NS3蛋白酶的变构抑制剂,在小鼠模型中具有口服疗效。

Ontoria, Jesus M; Torrente, Esther; Missineo, Antonino; Alli, Cristina; Graziani, Rita; Conti, Silvia; Bisbocci, Monica; Quotadamo, Antonio; Ferrigno, Federica; Corio, Alessandra; Ievoli, Giovanni; Bencheva, Leda; Amaudrut, Jérôme; Vasile, Silvana; Beghetto, Elisa; Paolini, Chantal; Alaimo, Nadine; Veneziano, Maria; Nibbio, Martina; Orsale, Maria V; Proto, Giulia; Colaceci, Fabrizio; Orsatti, Laura; Pucci, Vincenzo; Di Fabio, Romano; Tomei, Licia; Montalbetti, Christian; Bresciani, Alberto; Toniatti, Carlo; Paonessa, Giacomo

A phenotypic screen for novel small molecules that correct tau-mediated pathologies in human frontotemporal dementia neurons.

对能够纠正人类额颞叶痴呆神经元中 tau 蛋白介导的病理的新型小分子进行表型筛选

Maxwell Hannah, Smith James, Campbell Tom, Clark Jason, La Rocca Rosanna, Paonessa Francesco, Sitnikov Sergey, Evans Mark, Maycox Peter, Livesey Frederick J

The Bee Gut Microbiota: Bridging Infective Agents Potential in the One Health Context.

蜜蜂肠道微生物群:在一体化健康背景下连接感染因子的潜力

Tilocca Bruno, Greco Viviana, Piras Cristian, Ceniti Carlotta, Paonessa Mariachiara, Musella Vincenzo, Bava Roberto, Palma Ernesto, Morittu Valeria Maria, Spina Anna Antonella, Castagna Fabio, Urbani Andrea, Britti Domenico, Roncada Paola

Acute compartment syndrome and fasciotomy after a viper bite in Italy: a case report

意大利一例蝰蛇咬伤后急性筋膜室综合征及筋膜切开术病例报告

Sassoè-Pognetto, Marco; Cavalcante, Riccardo; Paonessa, Matteo

Synchronisation of apical constriction and cell cycle progression is a conserved behaviour of pseudostratified neuroepithelia informed by their tissue geometry

顶端收缩和细胞周期进程的同步是假复层神经上皮的保守行为,由其组织几何形状决定

Ioakeim Ampartzidis, Christoforos Efstathiou, Francesco Paonessa, Elliott M Thompson, Tyler Wilson, Conor J McCann, Nicholas DE Greene, Andrew J Copp, Frederick J Livesey, Nicola Elvassore, Giovanni G Giobbe, Paolo De Coppi, Eirini Maniou, Gabriel L Galea

Gametocyte-specific and all-blood-stage transmission-blocking chemotypes discovered from high throughput screening on Plasmodium falciparum gametocytes

通过对恶性疟原虫配子体进行高通量筛选发现配子体特异性和全血液阶段传播阻断化学型

Giacomo Paonessa #, Giulia Siciliano #, Rita Graziani, Cristiana Lalli, Ottavia Cecchetti, Cristina Alli, Roberto La Valle, Alessia Petrocchi, Alessio Sferrazza, Monica Bisbocci, Mario Falchi, Carlo Toniatti, Alberto Bresciani, Pietro Alano

Spiro-containing derivatives show antiparasitic activity against Trypanosoma brucei through inhibition of the trypanothione reductase enzyme

含螺环的衍生物通过抑制锥虫硫酮还原酶表现出对布氏锥虫的抗寄生虫活性

Lorenzo Turcano, Theo Battista, Esther Torrente De Haro, Antonino Missineo, Cristina Alli, Giacomo Paonessa, Gianni Colotti, Steven Harper, Annarita Fiorillo, Andrea Ilari, Alberto Bresciani

Microtubules Deform the Nuclear Membrane and Disrupt Nucleocytoplasmic Transport in Tau-Mediated Frontotemporal Dementia

在 Tau 介导的额颞叶痴呆症中,微管使核膜变形并破坏核质运输

Francesco Paonessa, Lewis D Evans, Ravi Solanki, Delphine Larrieu, Selina Wray, John Hardy, Stephen P Jackson, Frederick J Livesey

Latin America and the Caribbean Code Against Cancer: Developing Evidence-Based Recommendations to Reduce the Risk of Cancer in Latin America and the Caribbean

拉丁美洲和加勒比地区抗癌准则:制定循证建议以降低拉丁美洲和加勒比地区的癌症风险

Cazap, Eduardo; de Almeida, Liz Maria; Arrossi, Silvina; García, Patricia J; Garmendia, María Luisa; Gil, Enrique; Hassel, Trevor; Mayorga, Rubén; Mohar, Alejandro; Murillo, Raúl; Owen, Gabriel O; Paonessa, Diego; Santamaría, Julio; Tortolero-Luna, Guillermo; Zoss, Walter; Herrero, Rolando; Luciani, Silvana; Schüz, Joachim; Espina, Carolina

Identification of novel multi-stage histone deacetylase (HDAC) inhibitors that impair Schistosoma mansoni viability and egg production

鉴定新型多阶段组蛋白去乙酰化酶 (HDAC) 抑制剂,以削弱曼氏血吸虫的生存能力和产卵量

Alessandra Guidi, Fulvio Saccoccia, Nadia Gennari, Roberto Gimmelli, Emanuela Nizi, Cristiana Lalli, Giacomo Paonessa, Giuliana Papoff, Alberto Bresciani, Giovina Ruberti