日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification and Validation of an Inhibitor of the Protein Kinases PIM and DYRK.

鉴定和验证蛋白激酶 PIM 和 DYRK 的抑制剂。

Bencze Gyula, Venkataramani Prabhadevi, Elkayam Elad, Rivera Keith D, Garg Ankur, Szabadakai Istvan, Orfi Laszlo, Joshua-Tor Leemor, Pappin Darryl J, Tonks Nicholas K

Dietary pro-oxidant therapy by a vitamin K precursor targets PI 3-kinase VPS34 function.

通过维生素 K 前体进行膳食促氧化疗法,可靶向 PI 3-激酶 VPS34 的功能

Swamynathan Manojit M, Kuang Shan, Watrud Kaitlin E, Doherty Mary R, Gineste Charlotte, Mathew Grinu, Gong Grace Q, Cox Hilary, Cheng Eileen, Reiss David, Kendall Jude, Ghosh Diya, Reczek Colleen R, Zhao Xiang, Herzka Tali, Špokaitė Saulė, Dessus Antoine N, Kim Seung Tea, Klingbeil Olaf, Liu Juan, Nowak Dawid G, Alsudani Habeeb, Wee Tse-Luen, Park Youngkyu, Minicozzi Francesca, Rivera Keith, Almeida Ana S, Chang Kenneth, Chakrabarty Ram P, Wilkinson John E, Gimotty Phyllis A, Diermeier Sarah D, Egeblad Mikala, Vakoc Christopher R, Locasale Jason W, Chandel Navdeep S, Janowitz Tobias, Hicks James B, Wigler Michael, Pappin Darryl J, Williams Roger L, Cifani Paolo, Tuveson David A, Laporte Jocelyn, Trotman Lloyd C

TIMP1 is an early biomarker for detection and prognosis of lung cancer

TIMP1是肺癌早期检测和预后的生物标志物。

Dantas, Ezequiel; Murthy, Anirudh; Ahmed, Tanvir; Ahmed, Mujmmail; Ramsamooj, Shakti; Hurd, Maurice A; Lam, Tiffany; Malbari, Murtaza; Agrusa, Christopher; Elemento, Olivier; Zhang, Chen; Pappin, Darryl J; McGraw, Timothy E; Stiles, Brendon M; Altorki, Nasser K; Goncalves, Marcus D

Prostate tumor-induced stromal reprogramming generates Tenascin C that promotes prostate cancer metastasis through YAP/TAZ inhibition

前列腺肿瘤诱导的基质重编程产生腱生蛋白C,后者通过抑制YAP/TAZ促进前列腺癌转移。

Lee, Yu-Chen; Lin, Song-Chang; Yu, Guoyu; Zhu, Ming; Song, Jian H; Rivera, Keith; Pappin, Darryl J; Logothetis, Christopher J; Panaretakis, Theocharis; Wang, Guocan; Yu-Lee, Li-Yuan; Lin, Sue-Hwa

Tryp-N: A Thermostable Protease for the Production of N-terminal Argininyl and Lysinyl Peptides

Tryp-N:一种用于生产N端精氨酰肽和赖氨酰肽的耐热蛋白酶

Wilson, John P; Ipsaro, Jonathan J; Del Giudice, Samantha N; Turna, Nikita Saha; Gauss, Carla M; Dusenbury, Katharine H; Marquart, Krisann; Rivera, Keith D; Pappin, Darryl J

The glycan CA19-9 promotes pancreatitis and pancreatic cancer in mice

糖链CA19-9可促进小鼠胰腺炎和胰腺癌的发生。

Engle, Dannielle D; Tiriac, Hervé; Rivera, Keith D; Pommier, Arnaud; Whalen, Sean; Oni, Tobiloba E; Alagesan, Brinda; Lee, Eun Jung; Yao, Melissa A; Lucito, Matthew S; Spielman, Benjamin; Da Silva, Brandon; Schoepfer, Christina; Wright, Kevin; Creighton, Brianna; Afinowicz, Lauren; Yu, Kenneth H; Grützmann, Robert; Aust, Daniela; Gimotty, Phyllis A; Pollard, Katherine S; Hruban, Ralph H; Goggins, Michael G; Pilarsky, Christian; Park, Youngkyu; Pappin, Darryl J; Hollingsworth, Michael A; Tuveson, David A

DPM-1001 decreased copper levels and ameliorated deficits in a mouse model of Wilson's disease

DPM-1001降低了小鼠威尔逊病模型中的铜水平并改善了其功能缺陷。

Krishnan, Navasona; Felice, Christy; Rivera, Keith; Pappin, Darryl J; Tonks, Nicholas K

Mitochondrial Complex I Inhibitors Expose a Vulnerability for Selective Killing of Pten-Null Cells

线粒体复合物 I 抑制剂暴露了选择性杀死 Pten 缺失细胞的脆弱性

Naguib, Adam; Mathew, Grinu; Reczek, Colleen R; Watrud, Kaitlin; Ambrico, Alexandra; Herzka, Tali; Salas, Irene Casanova; Lee, Matthew F; El-Amine, Nour; Zheng, Wu; Di Francesco, M Emilia; Marszalek, Joseph R; Pappin, Darryl J; Chandel, Navdeep S; Trotman, Lloyd C

Efficient Reassignment of a Frequent Serine Codon in Wild-Type Escherichia coli

高效重分配野生型大肠杆菌中频繁出现的丝氨酸密码子

Ho, Joanne M; Reynolds, Noah M; Rivera, Keith; Connolly, Morgan; Guo, Li-Tao; Ling, Jiqiang; Pappin, Darryl J; Church, George M; Söll, Dieter

NSD3-Short Is an Adaptor Protein that Couples BRD4 to the CHD8 Chromatin Remodeler

NSD3-Short 是一种衔接蛋白,可将 BRD4 与 CHD8 染色质重塑因子偶联。

Shen, Chen; Ipsaro, Jonathan J; Shi, Junwei; Milazzo, Joseph P; Wang, Eric; Roe, Jae-Seok; Suzuki, Yutaka; Pappin, Darryl J; Joshua-Tor, Leemor; Vakoc, Christopher R