Fragment-Based Drug Design of Novel Pyranopyridones as Cell Active and Orally Bioavailable Tankyrase Inhibitors
基于片段的新型吡喃并吡啶酮类化合物药物设计:具有细胞活性和口服生物利用度的Tankyrase抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5b00251
de Vicente, Javier; Tivitmahaisoon, Parcharee; Berry, Pamela; Bolin, David R; Carvajal, Daisy; He, Wei; Huang, Kuo-Sen; Janson, Cheryl; Liang, Lena; Lukacs, Christine; Petersen, Ann; Qian, Hong; Yi, Lin; Zhuang, Yong; Hermann, Johannes C