日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

FDA Approval Summary: Mirvetuximab Soravtansine-Gynx for FRα-Positive, Platinum-Resistant Ovarian Cancer

FDA批准摘要:Mirvetuximab Soravtansine-Gynx用于治疗FRα阳性、铂类耐药卵巢癌

Dilawari, Asma; Shah, Mirat; Ison, Gwynn; Gittleman, Haley; Fiero, Mallorie H; Shah, Ankit; Hamed, Salaheldin S; Qiu, Junshan; Yu, Jingyu; Manheng, Wimolnut; Ricks, Tiffany K; Pragani, Rajan; Arudchandran, Arulvathani; Patel, Paresma; Zaman, Shadia; Roy, Arpita; Kalavar, Shyam; Ghosh, Soma; Pierce, William F; Rahman, Nam Atiqur; Tang, Shenghui; Mixter, Bronwyn D; Kluetz, Paul G; Pazdur, Richard; Amiri-Kordestani, Laleh

Patients experiences of their relationships with relatives and their collaboration with nurses during contact in non-COVID-19 hospital wards – A qualitative study

患者在非新冠肺炎病房与亲属接触期间与护士合作的经历——一项定性研究

Przepiorka, Donna; Le, Robert Q; Ionan, Alexei; Li, Ruo-Jing; Wang, Ying-Hong; Gudi, Ramadevi; Mitra, Soumya; Vallejo, Jonathon; Okusanya, Olanrewaju O; Ma, Lian; Yang, Yuching; Patel, Paresma; Mezaache, Djelila; Shah, Rakhi; Banerjee, Anamitro; McLamore, Sherita; Maung, Adam N; Goldberg, Kirsten B; Pazdur, Richard; Theoret, Marc R; De Claro, R Angelo; Pedersen, Birgith; Lerbæk, Birgitte; Jørgensen, Lone; Haslund-Thomsen, Helle; Thorup, Charlotte Brun; Albrechtsen, Maja Thomsen; Jacobsen, Sara; Nielsen, Marie Germund; Kusk, Kathrine Hoffmann; Laugesen, Britt; Voldbjerg, Siri Lygum; Grønkjær, Mette; Bundgaard, Karin

Target Deconvolution of a Multikinase Inhibitor with Antimetastatic Properties Identifies TAOK3 as a Key Contributor to a Cancer Stem Cell-Like Phenotype

具有抗转移特性的多激酶抑制剂的靶标反卷积确定 TAOK3 是癌症干细胞样表型的关键因素

Yansong Bian #, Yaroslav Teper #, Lesley A Mathews Griner #, Taylor J Aiken, Vivek Shukla, Rajarshi Guha, Paul Shinn, Hong-Wu Xin, Holger Pflicke, Astin S Powers, Dandan Li, Jian-Kang Jiang, Paresma Patel, Steven A Rogers, Jeffrey Aubé, Marc Ferrer, Craig J Thomas, Udo Rudloff

Discovery of 3-(4-sulfamoylnaphthyl)pyrazolo[1,5-a]pyrimidines as potent and selective ALK2 inhibitors

发现 3-(4-氨磺酰基萘基)吡唑并[1,5-a]嘧啶类化合物是高效且选择性的 ALK2 抑制剂

Jiang, Jian-Kang; Huang, Xiuli; Shamim, Khalida; Patel, Paresma R; Lee, Arthur; Wang, Amy Q; Nguyen, Kimloan; Tawa, Gregory; Cuny, Gregory D; Yu, Paul B; Zheng, Wei; Xu, Xin; Sanderson, Philip; Huang, Wenwei

Efficient Synthesis of 1,9-Substituted Benzo[h][1,6]naphthyridin-2(1H)-ones and Evaluation of their Plasmodium falciparum Gametocytocidal Activities

高效合成1,9-取代苯并[h][1,6]萘啶-2(1H)-酮及其对恶性疟原虫配子体的杀灭活性评价

Li, Hao; Sun, Wei; Huang, Xiuli; Lu, Xiao; Patel, Paresma R; Kim, Myunghoon; Orr, Meghan J; Fisher, Richard M; Tanaka, Takeshi Q; McKew, John C; Simeonov, Anton; Sanderson, Philip E; Zheng, Wei; Williamson, Kim C; Huang, Wenwei

Anticancer Effects of Mesothelin-Targeted Immunotoxin Therapy Are Regulated by Tyrosine Kinase DDR1

间皮素靶向免疫毒素疗法的抗癌作用受酪氨酸激酶DDR1调控

Ali-Rahmani, Fatima; FitzGerald, David J; Martin, Scott; Patel, Paresma; Prunotto, Marco; Ormanoglu, Pinar; Thomas, Craig; Pastan, Ira

In vitro evaluation of imidazo[4,5-c]quinolin-2-ones as gametocytocidal antimalarial agents

体外评价咪唑并[4,5-c]喹啉-2-酮类药物作为配子体杀灭抗疟药的活性

Patel, Paresma R; Sun, Wei; Kim, Myunghoon; Huang, Xiuli; Sanderson, Philip E; Tanaka, Takeshi Q; McKew, John C; Simeonov, Anton; Williamson, Kim C; Zheng, Wei; Huang, Wenwei

Blocking downstream signaling pathways in the context of HDAC inhibition promotes apoptosis preferentially in cells harboring mutant Ras

在 HDAC 抑制的背景下阻断下游信号通路优先促进含有突变 Ras 的细胞凋亡

Julian C Bahr, Robert W Robey, Victoria Luchenko, Agnes Basseville, Arup R Chakraborty, Hanna Kozlowski, Gary T Pauly, Paresma Patel, Joel P Schneider, Michael M Gottesman, Susan E Bates

High-throughput matrix screening identifies synergistic and antagonistic antimalarial drug combinations

高通量基质筛选确定了协同和拮抗抗疟药物组合

Bryan T Mott, Richard T Eastman, Rajarshi Guha, Katy S Sherlach, Amila Siriwardana, Paul Shinn, Crystal McKnight, Sam Michael, Norinne Lacerda-Queiroz, Paresma R Patel, Pwint Khine, Hongmao Sun, Monica Kasbekar, Nima Aghdam, Shaun D Fontaine, Dongbo Liu, Tim Mierzwa, Lesley A Mathews-Griner, Marc Fe

Ru-Based Z-Selective Metathesis Catalysts with Modified Cyclometalated Carbene Ligands

具有改性环金属化卡宾配体的钌基Z选择性复分解催化剂

Bronner, Sarah M; Herbert, Myles B; Patel, Paresma R; Marx, Vanessa M; Grubbs, Robert H