日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Repositioning HDAC Inhibitors for Glioma Treatment: Synthesis and Biological Evaluation

HDAC抑制剂在胶质瘤治疗中的应用:合成与生物学评价

Furtado, Luciana Costa; Waitman, Karoline de Barros; Silva, Nuno A T F; Gouvea, Leticia Marcelino; Kronenberger, Thales; Toledo, Mônica Franco Zannini Junqueira; Ferreira, Elthon Gois; Machado-Neto, João Agostinho; Kruyt, Frank A E; Parise Filho, Roberto; Costa-Lotufo, Letícia V

Capsaicin-Inspired Hydroxamate Hybrids as Selective HDAC6 Inhibitors with Antiproliferative Activity in Hematological Malignancies

辣椒素衍生的羟肟酸酯杂合物作为选择性 HDAC6 抑制剂,在血液恶性肿瘤中具有抗增殖活性

Gimenez Borges, Lara; Alves, Thais Nascimento de Oliveira; Vassiliades, Sandra Valeria; Carlos, Jorge Antonio Elias Godoy; Waitman, Karoline de Barros; Hilscher, Sebastian; Schutkowski, Mike; Sippl, Wolfgang; Tavares, Maurício Temotheo; Toledo, Monica Franco Zannini Junqueira; Costa-Lotufo, Letícia Veras; Kronenberger, Thales; Machado-Neto, João Agostinho; Parise-Filho, Roberto

Enhancing venetoclax efficacy in leukemia through association with HDAC inhibitors

通过与 HDAC 抑制剂联合使用增强维奈托克治疗白血病的疗效

Carlos, Jorge Antonio Elias Godoy; Tavares, Mauricio Temotheo; Lima, Keli; de Almeida, Larissa Costa; de Barros Waitman, Karoline; Costa-Lotufo, Leticia Veras; Parise-Filho, Roberto; Machado-Neto, João Agostinho

Dona Flor and her two husbands: Discovery of novel HDAC6/AKT2 inhibitors for myeloid cancer treatment

唐娜·弗洛尔和她的两位丈夫:发现用于治疗髓系癌症的新型HDAC6/AKT2抑制剂

Waitman, Karoline B; Martin, Holli-Joi; Carlos, Jorge A E G; Braga, Rodolpho C; Souza, Vinícius A M; Melo-Filho, Cleber C; Hilscher, Sebastian; Toledo, Mônica F Z J; Tavares, Maurício T; Costa-Lotufo, Letícia V; Machado-Neto, João A; Schutkowski, Mike; Sippl, Wolfgang; Kronenberger, Thales; Alves, Vinicius M; Parise-Filho, Roberto; Muratov, Eugene N

Hybrid histone deacetylase-kinase inhibitor potentiates venetoclax-induced cell death in chronic lymphocytic leukemia

混合型组蛋白去乙酰化酶-激酶抑制剂可增强维奈托克诱导的慢性淋巴细胞白血病细胞死亡。

Garnique, Anali Del Milagro Bernabe; Carlos, Jorge Antonio Elias Godoy; Parducci, Natalia Sudan; Tavares, Mauricio Temotheo; Waitman, Karoline de Barros; Lima, Keli; Costa-Lotufo, Leticia Veras; Parise-Filho, Roberto; Machado-Neto, João Agostinho

Drug repositioning in the COVID-19 pandemic: fundamentals, synthetic routes, and overview of clinical studies

新冠疫情下的药物重定位:基本原理、合成路线和临床研究概述

Vaz, Elisa Souza; Vassiliades, Sandra Valeria; Giarolla, Jeanine; Polli, Michelle Carneiro; Parise-Filho, Roberto

Peppers: A "Hot" Natural Source for Antitumor Compounds

辣椒:一种富含抗肿瘤化合物的“辛辣”天然来源

Cunha, Micael Rodrigues; Tavares, Maurício Temotheo; Fernandes, Thais Batista; Parise-Filho, Roberto

Another Reason for Using Caffeine in Dermocosmetics: Sunscreen Adjuvant

在皮肤化妆品中使用咖啡因的另一个原因:防晒辅助剂

Rosado, Catarina; Tokunaga, Viviane Kaori; Sauce, Rafael; de Oliveira, Camila Areias; Sarruf, Fernanda Daud; Parise-Filho, Roberto; Maurício, Elisabete; de Almeida, Tânia Santos; Velasco, Maria Valéria Robles; Baby, André Rolim