GPCR Agonist-to-Antagonist Conversion: Enabling the Design of Nucleoside Functional Switches for the A(2A) Adenosine Receptor
GPCR激动剂到拮抗剂的转换:实现A(2A)腺苷受体核苷功能开关的设计
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.2c00462
Shiriaeva, Anna; Park, Daejin; Kim, Gyudong; Lee, Yoonji; Hou, Xiyan; Jarhad, Dnyandev B; Kim, Gibae; Yu, Jinha; Hyun, Young Eum; Kim, Woomi; Gao, Zhan-Guo; Jacobson, Kenneth A; Han, Gye Won; Stevens, Raymond C; Jeong, Lak Shin; Choi, Sun; Cherezov, Vadim