Discovery of MK-7145, an Oral Small Molecule ROMK Inhibitor for the Treatment of Hypertension and Heart Failure
发现MK-7145,一种用于治疗高血压和心力衰竭的口服小分子ROMK抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.6b00122
Tang, Haifeng; Zhu, Yuping; Teumelsan, Nardos; Walsh, Shawn P; Shahripour, Aurash; Priest, Birgit T; Swensen, Andrew M; Felix, John P; Brochu, Richard M; Bailey, Timothy; Thomas-Fowlkes, Brande; Pai, Lee-Yuh; Hampton, Caryn; Corona, Aaron; Hernandez, Melba; Metzger, Joseph; Forrest, Michael; Zhou, Xiaoyan; Owens, Karen; Tong, Vincent; Parmee, Emma; Roy, Sophie; Kaczorowski, Gregory J; Yang, Lihu; Alonso-Galicia, Magdalena; Garcia, Maria L; Pasternak, Alexander