日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Xanomeline treatment attenuates cocaine self-administration in rats and nonhuman primates

Xanomeline治疗可减轻大鼠和非人灵长类动物的可卡因自我给药行为。

Marsh, Samuel A; Heslep, Nicholas; Paronis, Carol A; Bergman, Jack; Negus, S Stevens; Banks, Matthew L

The Effects of Chronic Naltrexone on Reinstatement of Opioid-Induced Drug-Seeking Behavior and Antinociception

长期服用纳曲酮对阿片类药物诱发的觅药行为恢复和镇痛作用的影响

Withey, Sarah L; Bergman, Jack; Paronis, Carol A

Effects of inhaled low-concentration xenon gas on naltrexone-precipitated withdrawal symptoms in morphine-dependent mice

吸入低浓度氙气对吗啡依赖小鼠纳曲酮诱发戒断症状的影响

Kaufman, Marc J; Meloni, Edward G; Qrareya, Alaa N; Paronis, Carol A; Bogin, Vlad

Ole-Oxy, a Semi-Synthetic Analog of Oleuropein, Ameliorates Acute Skin and Colon Inflammation in Mice

Ole-Oxy 是橄榄苦苷的半合成类似物,可改善小鼠的急性皮肤和结肠炎症

Nikolaos V Angelis, Efthymios Paronis, Georgia Sarikaki, Antonios Kyriakopoulos, Anna Agapaki, Pigi-Maria Niotopoulou, Christina C Knai, Pavlos Alexakos, Odyssefs Liagkas, Konstantinos F Mavreas, Constantin N Baxevanis, Alexios-Leandros Skaltsounis, Ourania E Tsitsilonis, Ioannis K Kostakis

Discovery of a Potent Highly Biased MOR Partial Agonist among Diastereomeric C9-Hydroxyalkyl-5-phenylmorphans

在非对映异构体 C9-羟烷基-5-苯基吗啡烷中发现一种强效高偏向性 MOR 部分激动剂

Lutz, Joshua A; Sulima, Agnieszka; Gutman, Eugene S; Bow, Eric W; Luo, Dan; Kaska, Sophia; Prisinzano, Thomas E; Paronis, Carol A; Bergman, Jack; Imler, Gregory H; Kerr, Andrew T; Jacobson, Arthur E; Rice, Kenner C

Supplementation with uric and ascorbic acid protects stored red blood cells through enhancement of non-enzymatic antioxidant activity and metabolic rewiring

补充尿酸和抗坏血酸可通过增强非酶抗氧化活性和代谢重组来保护储存的红细胞

Vassilis L Tzounakas, Alkmini T Anastasiadi, Vasiliki-Zoi Arvaniti, Veronica Lelli, Giuseppina Fanelli, Efthymios C Paronis, Anastasia C Apostolidou, Evangelos G Balafas, Nikolaos G Kostomitsopoulos, Effie G Papageorgiou, Issidora S Papassideri, Konstantinos Stamoulis, Anastasios G Kriebardis, Sara

A Journey through Diastereomeric Space: The Design, Synthesis, In Vitro and In Vivo Pharmacological Activity, and Molecular Modeling of Novel Potent Diastereomeric MOR Agonists and Antagonists

非对映异构体空间之旅:新型高效非对映异构体MOR激动剂和拮抗剂的设计、合成、体外和体内药理活性及分子建模

Chambers, Dana R; Sulima, Agnieszka; Luo, Dan; Prisinzano, Thomas E; Goldberg, Alexander; Xie, Bing; Shi, Lei; Paronis, Carol A; Bergman, Jack; Nassehi, Nima; Selley, Dana E; Imler, Gregory H; Jacobson, Arthur E; Rice, Kenner C

NLX-112, a highly selective 5-HT(1A) receptor biased agonist, does not exhibit misuse potential in male rats or macaques

NLX-112 是一种高选择性的 5-HT(1A) 受体偏向性激动剂,在雄性大鼠或猕猴中未表现出滥用潜力。

Depoortère, R; Bergman, J; Beardsley, P M; Desai, R I; Paronis, C A; Walentiny, D M; Varney, M A; Newman-Tancredi, A

Corpuscular Fragility and Metabolic Aspects of Freshly Drawn Beta-Thalassemia Minor RBCs Impact Their Physiology and Performance Post Transfusion: A Triangular Correlation Analysis In Vitro and In Vivo

新鲜采集的β-地中海贫血轻型红细胞的细胞脆性和代谢特性影响其输血后的生理和功能:体外和体内三角相关性分析

Anastasiadi, Alkmini T; Arvaniti, Vasiliki-Zoi; Paronis, Efthymios C; Kostomitsopoulos, Nikolaos G; Stamoulis, Konstantinos; Papassideri, Issidora S; D'Alessandro, Angelo; Kriebardis, Anastasios G; Tzounakas, Vassilis L; Antonelou, Marianna H

Altered sleep during spontaneous cannabinoid withdrawal in male mice

雄性小鼠自发性戒断大麻素期间睡眠改变

Missig, Galen; Mehta, Niyati; Robbins, James O; Good, Cameron H; Iliopoulos-Tsoutsouvas, Christos; Makriyannis, Alex; Nikas, Spyros P; Bergman, Jack; Carlezon, William A Jr; Paronis, Carol A