Discovery of κ Opioid Receptor (KOR)-Selective d-Tetrapeptides with Improved In Vivo Antinociceptive Effect after Peripheral Administration
发现具有增强的κ阿片受体(KOR)选择性d-四肽,其外周给药后体内镇痛作用增强
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.2c00237
Stefanucci, Azzurra; Della Valle, Alice; Scioli, Giuseppe; Marinaccio, Lorenza; Pieretti, Stefano; Minosi, Paola; Szucs, Edina; Benyhe, Sandor; Masci, Domiziana; Tanguturi, Parthasaradhireddy; Chou, Kerry; Barlow, Deborah; Houseknecht, Karen; Streicher, John M; Mollica, Adriano