日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and Biological Evaluation of Novel Acetylcholinesterase and β-Secretase 1 Inhibitors

新型乙酰胆碱酯酶和β-分泌酶1抑制剂的设计、合成及生物学评价

Drozdowska, Danuta; Pawelski, Damian; Wróbel-Tałałaj, Agnieszka; Plonska-Brzezinska, Marta; Kolesinska, Beata; Lazny, Ryszard; Seroka, Barbara; Parzych, Cezary; Ratkiewicz, Artur

Substituent and Ring-Number Effects on the Kinetics of PAH + OH Reactions: A QSAR-DOE Approach with Tunneling Corrections

取代基和环数对PAH + OH反应动力学的影响:基于隧道效应校正的QSAR-DOE方法

Parzych, Cezary; Baradyn, Maciej; Ratkiewicz, Artur

Rational design, synthesis, and molecular modelling insights of dual DNA binders/DHFR inhibitors bearing arylidene-hydrazinyl-1,3-thiazole scaffold with apoptotic and anti-migratory potential in breast MCF-7 cancer cells.

对具有亚芳基肼基-1,3-噻唑骨架的双重DNA结合剂/DHFR抑制剂进行合理设计、合成和分子建模,以研究其在乳腺癌MCF-7细胞中的凋亡和抗迁移潜力

El-Wakil Marwa H, Ghazala Rasha A, El-Dershaby Hadeel A, Drozdowska Danuta, Wróbel-Tałałaj Agnieszka, Parzych Cezary, Ratkiewicz Artur, Kolesińska Beata, Abd El-Razik Heba A, Soliman Farid S G

Repurposed Arylidene-hydrazinyl-1,3-thiazoles as Multitarget Anti-Alzheimer's Agents via Combined Computational and Experimental Studies

通过计算和实验相结合的研究,将亚芳基肼基-1,3-噻唑类化合物重新用于多靶点抗阿尔茨海默病治疗

Drozdowska, Danuta; Ratkiewicz, Artur; Wróbel-Tałałaj, Agnieszka; Parzych, Cezary; El-Dershaby, Hadeel A; Abd El-Razik, Heba A; Soliman, Farid S G; El-Wakil, Marwa H

Benzamide Trimethoprim Derivatives as Human Dihydrofolate Reductase Inhibitors-Molecular Modeling and In Vitro Activity Study

苯甲酰胺类甲氧苄啶衍生物作为人二氢叶酸还原酶抑制剂——分子建模和体外活性研究

Drozdowska, Danuta; Wróbel-Tałałaj, Agnieszka; Parzych, Cezary; Ratkiewicz, Artur