Highly Selective, Reversible Inhibitor Identified by Comparative Chemoproteomics Modulates Diacylglycerol Lipase Activity in Neurons
通过比较化学蛋白质组学鉴定出的高选择性、可逆抑制剂可调节神经元中的二酰甘油脂肪酶活性
期刊:Journal of the American Chemical Society
影响因子:15.6
doi:10.1021/jacs.5b04883
Baggelaar, Marc P; Chameau, Pascal J P; Kantae, Vasudev; Hummel, Jessica; Hsu, Ku-Lung; Janssen, Freek; van der Wel, Tom; Soethoudt, Marjolein; Deng, Hui; den Dulk, Hans; Allarà, Marco; Florea, Bogdan I; Di Marzo, Vincenzo; Wadman, Wytse J; Kruse, Chris G; Overkleeft, Herman S; Hankemeier, Thomas; Werkman, Taco R; Cravatt, Benjamin F; van der Stelt, Mario