日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Stereodefined Synthesis of 3-Difluoromethyl-Benzoxaboroles: Novel Antimicrobials with Unlocked H-Bonding

3-二氟甲基苯并硼氧杂环的立体定向合成:具有开放氢键的新型抗菌剂

Dimasi, Alessandro; Montoli, Arianna; Lutti, Claudio; Citarella, Andrea; Ronchi, Paolo; Castagnini, Francesco; Mileo, Valentina; Macetti, Giovanni; Baldelli, Valerio; Rossi, Elio; Landini, Paolo; Passarella, Daniele; Fasano, Valerio

Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer.

基于结构的Hsp90/HDAC6双重抑制剂的发现及其在侵袭性前列腺癌中的应用

Citarella Andrea, Belluti Silvia, Bonanni Davide, Moi Davide, Piccinini Isabella, Rinaldi Arianna, Papulino Chiara, Benedetti Rosaria, Cuoghi Laura, Ciolo Stefano Di, Silvani Alessandra, Altucci Lucia, Pinzi Luca, Franchini Silvia, Passarella Daniele, Sorbi Claudia, Giannini Clelia, Imbriano Carol, Rastelli Giulio

Sustainable Synthesis of 1,2,3-Triazoles using Cyrene as a Biodegradable Solvent in Click Chemistry

利用环己烯作为可生物降解溶剂,在点击化学中可持续合成1,2,3-三唑

Citarella, Andrea; Fiori, Alessandro; Silvani, Alessandra; Passarella, Daniele; Fasano, Valerio

Self-Assembled Cannabigerol-Based Nanoparticles: Design, Synthesis, and Antiproliferative Activity.

自组装大麻酚基纳米粒子:设计、合成和抗增殖活性

Amenta Arianna, Nordio Giulia, Piazzola Francesco, Di Paolo Maria Luisa, Milani Fabio, Giacomini Martina, Citarella Andrea, Ciriello Umberto, Paladino Giuseppe, Pellegrino Sara, Silvestri Federica, Fasano Valerio, Dalla Via Lisa, Passarella Daniele

Rotational Motion in Bispidines: A Conformational Study

双吡啶的旋转运动:构象研究

Migliano, Francesco; Pozzi, Luca; Citarella, Andrea; Macetti, Giovanni; Lo Presti, Leonardo; Passarella, Daniele; Fasano, Valerio

Automated fluorine-18 radiolabeling via an alkyne-azide cycloaddition reaction on a dual peptide-functionalized liposome surface for in vivo PET imaging

利用炔烃-叠氮环加成反应在双肽功能化脂质体表面进行自动化氟-18放射性标记,用于体内PET成像

Iannone, Marco; Kravicz, Marcelo; Rainone, Paolo; Antoniou, Antonia I; Stucchi, Stefano; Valtorta, Silvia; Amenta, Arianna; Turolla, Elia Anna; Pellegrino, Sara; Passarella, Daniele; Vino, Elisa; Todde, Sergio; Re, Francesca; Seneci, Pierfausto; Moresco, Rosa Maria

Mechanistic insights into the base-mediated deuteration of pyridyl phosphonium and ammonium salts

碱介导的吡啶基膦和铵盐氘代反应的机理研究

Montoli, Arianna; Dimasi, Alessandro; Guarnaccia, Miriana; Citarella, Andrea; Ronchi, Paolo; Blasi, Delia; Rossi, Sergio; Passarella, Daniele; Fasano, Valerio

Asymmetric Total Synthesis of (-)-Glycybridin B, a Pharmacophore Screened Candidate for Tubulin Binding

(-)-Glycybridin B 的不对称全合成,一种筛选出的微管蛋白结合药效团候选物

Maiocchi, Alice; Shevelev, Maxim; Boiarska, Zlata; Estévez-Gallego, Juan; Bonato, Francesca; Orlando, Paolo; Chinosi, Alessandra; Marcone, Emanuele; Citarella, Andrea; Horvath, Dragos; Steinmetz, Michel O; Prota, Andrea E; Varnek, Alexandre; Fasano, Valerio; Passarella, Daniele

Cannabizetol, a Novel Cannabinoid: Chemical Synthesis, Anti-inflammatory Activity and Extraction from Cannabis sativa L

大麻素Cannabizetol:化学合成、抗炎活性及从大麻(Cannabis sativa L.)中提取

Pozzi, Luca; Gotti, Andrea; Fumagalli, Marco; Citarella, Andrea; Fasano, Valerio; Paladino, Giuseppe; Ciriello, Umberto; Princiotto, Salvatore; Annunziata, Francesca; Martinelli, Giulia; Sangiovanni, Enrico; Pinto, Andrea; Dell'Agli, Mario; Passarella, Daniele

Cu-Catalyzed Asymmetric Synthesis of γ-Amino Alcohols Featuring Tertiary Carbon Stereocenters

铜催化不对称合成具有叔碳立体中心的γ-氨基醇

Delgado, Alejandro; Orlando, Paolo; Lanzi, Matteo; Benet-Buchholz, Jordi; Passarella, Daniele; Kleij, Arjan W