日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Pharmacology of a Morphinan-Derived Dual Mu-Kappa Opioid Receptor Agonist Analgesic.

吗啡烷衍生的双重μ-κ阿片受体激动剂镇痛药的合成与药理学研究

Varga Balazs R, Uprety Rajendra, Paul Barnali, Knoll Alexis, Ramos-Gonzalez Nokomis, Appourchaux Kevin, Taylor Tori, Turgutalp Bengisu, Shinouchi Ryosuke, Eans Shainnel O, Williams Ashai K, Vasquez-Grinnell Steven G, Zaidi Saheem, Nazarova Antonina L, Varadi Andras, Le Rouzic Valerie, Brown Taylor G, Martinez Shani, Ansonoff Michael, Dardashti Rebecca Notis, Hunkele Amanda, Subrath Joan, Welch Matthew, Xu Jin, Rossi Grace C, Pintar John, Pasternak Gavril W, Katritch Vsevolod, McLaughlin Jay P, Pan Ying Xian, Majumdar Susruta

Correction to: Mu Opioids Induce Biased Signaling at the Full-Length Seven Transmembrane C-Terminal Splice Variants of the mu Opioid Receptor Gene, Oprm1

更正:μ阿片受体在μ阿片受体基因Oprm1的全长七次跨膜C端剪接变体处诱导偏向性信号传导

Narayan, Ankita; Hunkele, Amanda; Xu, Jin; Bassoni, Daniel L; Pasternak, Gavril W; Pan, Ying-Xian

Confronting the opioid crisis with basic research in neuropharmacology

利用神经药理学基础研究应对阿片类药物危机

Baumann, Michael H; Pasternak, Gavril W; Negus, Sidney S

7-Hydroxymitragynine Is an Active Metabolite of Mitragynine and a Key Mediator of Its Analgesic Effects

7-羟基帽柱木碱是帽柱木碱的活性代谢产物,也是其镇痛作用的关键介质。

Kruegel, Andrew C; Uprety, Rajendra; Grinnell, Steven G; Langreck, Cory; Pekarskaya, Elizabeth A; Le Rouzic, Valerie; Ansonoff, Michael; Gassaway, Madalee M; Pintar, John E; Pasternak, Gavril W; Javitch, Jonathan A; Majumdar, Susruta; Sames, Dalibor

MP1104, a mixed kappa-delta opioid receptor agonist has anti-cocaine properties with reduced side-effects in rats

MP1104是一种混合型κ-δ阿片受体激动剂,具有抗可卡因特性,且在大鼠中副作用较小。

Atigari, Diana V; Uprety, Rajendra; Pasternak, Gavril W; Majumdar, Susruta; Kivell, Bronwyn M

Pharmacological Characterization of Levorphanol, a G-Protein Biased Opioid Analgesic

左吗啡醇(一种G蛋白偏向性阿片类镇痛药)的药理学特征

Le Rouzic, Valerie; Narayan, Ankita; Hunkle, Amanda; Marrone, Gina F; Lu, Zhigang; Majumdar, Susruta; Xu, Jin; Pan, Ying-Xian; Pasternak, Gavril W

Significance of the Stress Research: “In Memoriam, Richard Kvetnansky”

压力研究的意义:“纪念理查德·克维特南斯基”

Sudduth-Klinger, J; Schumann, M; Gardner, P; Payan, D G; Childers, Steven R; Pasternak, Gavril W; Biondi, Carla; Belardetti, Francesco; Brunelli, Marcello; Portolan, Alice; Trevisani, Agostino; Dimpfel, Wilfried; Briggs, Clark A; Whiting, Gary J; Ariano, Marjorie A; McAfee, Donald A; Partridge, L Donald; Osborne, N N; Beale, R; Nicholas, D; Stadler, H; Walker, J H; Jones, R T; Whittaker, V P; Chesnut, Thomas J; Grewe, C W; Kebabian, J W; Saavedra, J M; Barden, N; Chevillard, C; Fernandez-Pardal, J; Shtark, M B; Tretyakov, V P; Deriy, B N; Zapara, T A; Carpenter, David O; Raizada, Mohan K; Stamler, John F; Quinlan, James T; Landas, Steve; Phillips, M Ian; Saavedra, Juan M; Saavedra, Juan M; Creveling, C R; Deli, Ma’ria A; Nabika, Toru; Yamori, Yukio; Saavedra, Juan M; Carpenter, David O; Dubocovich, Margarita L; Dubocovich, Margarita L; Slater, N T; Carpenter, D O; Ariano, Marjorie A; Briggs, Clark A; McAfee, Donald A; Petrunyaka, V V; Bowen, Wayne D; Pert, Candace B; Haas, H L; Felix, D; Davis, M D; Galli, Daniela; De Nicola, Alejandro F; de Vellis, Jean; Libertun, Carlos; Sakharov, Dmitri A; Croll, Roger P; Aréchiga, Hugo; Gainer, Harold; Libertun, Carlos; Aréchiga, Hugo; Gainer, Harold; Mohanakumar, K P; Saavedra, Juan M; Souza, Diogo O; Libertun, Carlos; De Nicola, Alejandro F; Gomez, Marcus Vinicius; Alexander, Kiss; Nikodémová, Mária; Kučerová, Jana; Štrbák, Vladimír; Talman, William T; Sved, Alan; Saunders, N R; Dziegielewska, K M; Eiden, Lee E; Paila, Yamuna Devi; Chattopadhyay, Amitabha; Saavedra, Juan M; Gerozissis, Kyriaki; Kato, Hiroyuki; Kogure, Kyuya; Lombardi, V; Valko, L; Valko, M; Scozzafava, A; Morris, H; Melnik, M; Svitel, J; Budešinský, M; Pelnár, J; Steno, J; Liptaj, T; Zalibera, L; Budinská, J; Zlatoš, J; Giuliani, A; Mascolo, L; Leibfritz, D; Murer, M G; Tseng, K Y; Kasanetz, F; Belluscio, M; Riquelme, L A; Champier, J; Jouvet, A; Rey, C; Guyotat, J; Fevre-Montange, M; Kvetnansky, Richard; Wang, Xueyu; Ma, Aihua; Zhu, Weiwei; Zhu, Liping; Zhao, Yutian; Xi, Jiashui; Zhang, Xinying; Zhao, Bojun; Lu, Lin; Fang, Yuxia; Wang, Xi; Saavedra, Juan M; Baker, Glen B; Saavedra, Juan M; Zorad, Stefan; Jezova, Daniela; Strbak, Vladimir; Macho, Ladislav; Saavedra, Juan M

Alternatively spliced mu opioid receptor C termini impact the diverse actions of morphine

μ阿片受体C端选择性剪接影响吗啡的多种作用

Xu, Jin; Lu, Zhigang; Narayan, Ankita; Le Rouzic, Valerie P; Xu, Mingming; Hunkele, Amanda; Brown, Taylor G; Hoefer, William F; Rossi, Grace C; Rice, Richard C; Martínez-Rivera, Arlene; Rajadhyaksha, Anjali M; Cartegni, Luca; Bassoni, Daniel L; Pasternak, Gavril W; Pan, Ying-Xian

Genetic dissociation of morphine analgesia from hyperalgesia in mice

小鼠吗啡镇痛作用与痛觉过敏的遗传分离

Marrone, Gina F; Le Rouzic, Valerie; Varadi, Andras; Xu, Jin; Rajadhyaksha, Anjali M; Majumdar, Susruta; Pan, Ying-Xian; Pasternak, Gavril W

Isolation and characterization of alternatively spliced variants of the mouse sigma1 receptor gene, Sigmar1

小鼠 sigma1 受体基因 Sigmar1 的选择性剪接变体的分离和鉴定

Pan, Ling; Pasternak, David A; Xu, Jin; Xu, Mingming; Lu, Zhigang; Pasternak, Gavril W; Pan, Ying-Xian