日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Single-position ligand modifications tune CB(2)R activity by targeting the toggle switch

通过靶向开关,单点配体修饰可以调节 CB(2)R 的活性。

Ganzoni, Rudolf L Z; Kosar, Miroslav; Han, Yongqi; Vitale, Rosa Maria; Amodeo, Pietro; Li, Xiaoting; Zha, Zhonghua; Patej, Kacper J; Kicin, Bilal; Strunden, Taddäus E N; Reichert, Lisa; Gómez-Bouzó, Uxía; Perera, Themiya P; Atz, Kenneth; Guba, Wolfgang; Bartelmus, Christian; Bigler, Raphael; Tosatti, Paolo; Bachmann, Stephan; Hua, Tian; Sykes, David A; Veprintsev, Dmitry B; Grether, Uwe; Carreira, Erick M

A universal cannabinoid CB1 and CB2 receptor TR-FRET kinetic ligand-binding assay.

一种通用的大麻素 CB1 和 CB2 受体 TR-FRET 动力学配体结合测定法

Borrega-Roman Leire, Hoare Bradley L, Kosar Miroslav, Sarott Roman C, Patej Kacper J, Bouma Jara, Scott-Dennis Morgan, Koers Eline J, Gazzi Thais, Mach Leonard, Barrondo Sergio, Sallés Joan, Guba Wolfgang, Kusznir Eric, Nazaré Marc, Rufer Arne C, Grether Uwe, Heitman Laura H, Carreira Erick M, Sykes David A, Veprintsev Dmitry B

Flipping the GPCR Switch: Structure-Based Development of Selective Cannabinoid Receptor 2 Inverse Agonists

翻转GPCR开关:基于结构的选择性大麻素受体2反向激动剂的开发

Kosar, Miroslav; Sarott, Roman C; Sykes, David A; Viray, Alexander E G; Vitale, Rosa Maria; Tomašević, Nataša; Li, Xiaoting; Ganzoni, Rudolf L Z; Kicin, Bilal; Reichert, Lisa; Patej, Kacper J; Gómez-Bouzó, Uxía; Guba, Wolfgang; McCormick, Peter J; Hua, Tian; Gruber, Christian W; Veprintsev, Dmitry B; Frank, James A; Grether, Uwe; Carreira, Erick M