日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Highly Sensitive Multiplexed Detection of Brain‐Derived Tau and Phosphorylated Tau Proteoforms with the NULISA Technology

利用NULISA技术对脑源性tau蛋白和磷酸化tau蛋白进行高灵敏度多重检测

Wang, Yi-Jun; Patel, Bhargav A; Anreddy, Nagaraju; Zhang, Yun-Kai; Zhang, Guan-Nan; Alqahtani, Saeed; Singh, Satyakam; Shukla, Suneet; Kaddoumi, Amal; Ambudkar, Suresh V; Talele, Tanaji T; Chen, Zhe-Sheng; Ma, Xiao‐Jun; Iyengar, Shweta; Deshmukh, Shalaka; Comandor, Roopa; Wang, Li; Kim, Sean; Xu, Xiaomei; Feng, Wei; Qiu, Xiaolei; Zhang, Bingqing; Luo, Yuling

Manassantin A inhibits tumour growth under hypoxia through the activation of chaperone-mediated autophagy by modulating Hsp90 activity

马纳桑汀A通过调节Hsp90活性激活分子伴侣介导的自噬,从而抑制缺氧条件下的肿瘤生长。

Byun, Jun-Kyu; Lee, Sun Hee; Moon, Eui Jung; Park, Myo-Hyeon; Jang, Hyeonha; Weitzel, Douglas H; Kim, Hyun-Hwi; Basnet, Nikita; Kwon, Do-Yeon; Lee, Chen-Ting; Stephenson, Tesia N; Jeong, Ji-Hak; Patel, Bhargav A; Park, Sung Jean; Chi, Jen-Tsan; Dewhirst, Mark W; Hong, Jiyong; Lee, You Mie

CryoEM Structure with ATP Synthase Enables Late-Stage Diversification of Cruentaren A

利用冷冻电镜技术解析ATP合成酶结构,揭示克鲁恩塔伦A后期多样化的机制

Dou, Xiaozheng; Guo, Hui; D'Amico, Terin; Abdallah, Leah; Subramanian, Chitra; Patel, Bhargav A; Cohen, Mark; Rubinstein, John L; Blagg, Brian S J

Natural products and other inhibitors of F(1)F(O) ATP synthase

天然产物和其他F(1)F(O) ATP合酶抑制剂

Patel, Bhargav A; D'Amico, Terin L; Blagg, Brian S J

Thiazole-valine peptidomimetic (TTT-28) antagonizes multidrug resistance in vitro and in vivo by selectively inhibiting the efflux activity of ABCB1

噻唑-缬氨酸肽模拟物(TTT-28)通过选择性抑制ABCB1的外排活性,在体外和体内拮抗多药耐药性。

Wang, Yi-Jun; Patel, Bhargav A; Anreddy, Nagaraju; Zhang, Yun-Kai; Zhang, Guan-Nan; Alqahtani, Saeed; Singh, Satyakam; Shukla, Suneet; Kaddoumi, Amal; Ambudkar, Suresh V; Talele, Tanaji T; Chen, Zhe-Sheng

Semi-synthetic ocotillol analogues as selective ABCB1-mediated drug resistance reversal agents.

半合成的奥可替洛尔类似物作为选择性 ABCB1 介导的耐药性逆转剂

Zhang Yun-Kai, Zhang Hengyuan, Zhang Guan-Nan, Wang Yi-Jun, Kathawala Rishil J, Si Rui, Patel Bhargav A, Xu Jinyi, Chen Zhe-Sheng

Design, synthesis, and biological evaluation of (S)-valine thiazole-derived cyclic and noncyclic peptidomimetic oligomers as modulators of human P-glycoprotein (ABCB1)

设计、合成和生物学评价(S)-缬氨酸噻唑衍生的环状和非环状肽模拟寡聚体作为人类P-糖蛋白(ABCB1)调节剂

Singh, Satyakam; Prasad, Nagarajan Rajendra; Kapoor, Khyati; Chufan, Eduardo E; Patel, Bhargav A; Ambudkar, Suresh V; Talele, Tanaji T

Design and synthesis of L- and D-phenylalanine derived rhodanines with novel C5-arylidenes as inhibitors of HCV NS5B polymerase

设计和合成以新型C5-亚芳基取代的L-和D-苯丙氨酸衍生的罗丹宁类化合物作为HCV NS5B聚合酶抑制剂

Patel, Bhargav A; Krishnan, Ramalingam; Khadtare, Nikhil; Gurukumar, K R; Basu, Amartya; Arora, Payal; Bhatt, Aaditya; Patel, Maulik R; Dana, Dibyendu; Kumar, Sanjai; Kaushik-Basu, Neerja; Talele, Tanaji T