日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacokinetic, Safety, and Pharmacodynamic Profiles of Saroglitazar Magnesium in Cholestatic Cirrhosis With Hepatic Impairment and Participants With Renal Impairment

沙格列汀镁在伴有肝功能损害的胆汁淤积性肝硬化患者和伴有肾功能损害的受试者中的药代动力学、安全性和药效学特征

Vuppalanchi, Raj; Cruz, Mary M; Momin, Taufik; Shaikh, Farheen; Swint, Kimberly; Patel, Harilal; Parmar, Deven

Prolyl hydroxylase inhibitor desidustat improves stroke outcomes via enhancing efferocytosis in mice with chronic kidney disease.

脯氨酰羟化酶抑制剂地西达司他通过增强慢性肾病小鼠的胞吞作用来改善中风预后

Kaur Harpreet, Pandey Nilesh, Chandaluri Lakshmi, Shaaban Nirvana, Martinez Alexa, Kidder Evan, Patel Vishal J, Kshirsagar Samadhan G, Kumar Dhananjay, Frausto Louise, Pandit Rajan, Richard Koral S E, Anand Sumit Kumar, Das Sandeep, Vikram Ajit, Magdy Tarek, Lu Xiao-Hong, Orr A Wayne, Patel Harilal, Trivedi Ravi Kumar, Kansagra Kevinkumar, Joharapurkar Amit A, Parmar Deven V, Jain Mukul R, Rom Oren, Yurdagul Arif Jr, Dhanesha Nirav

Desidustat: a novel PHD inhibitor for the treatment of CKD-induced anemia

Desidustat:一种用于治疗CKD相关贫血的新型PHD抑制剂

Joharapurkar, Amit; Pandya, Vrajesh; Patel, Harilal; Jain, Mukul; Desai, Ranjit

Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of the Oral NLRP3 Inflammasome Inhibitor ZYIL1: First-in-Human Phase 1 Studies (Single Ascending Dose and Multiple Ascending Dose)

口服 NLRP3 炎症小体抑制剂 ZYIL1 的安全性、耐受性、药代动力学和药效学:首次人体 1 期研究(单次递增剂量和多次递增剂量)

Parmar, Deven V; Kansagra, Kevinkumar A; Momin, Taufik; Patel, Hardik B; Jansari, Gaurav A; Bhavsar, Jay; Shah, Chintan; Patel, Jayesh M; Ghoghari, Ashok; Barot, Ajay; Sharma, Bhavesh; Viswanathan, Kasinath; Patel, Harilal V; Jain, Mukul R

Non-clinical safety evaluation of a novel pharmaceutical salt, rosuvastatin ethanolamine, in Wistar rats

在Wistar大鼠中对一种新型药物盐——瑞舒伐他汀乙醇胺进行非临床安全性评价

Vaghasiya, Jigneshkumar; Patel, Satyam; Patel, Sudhir; Kadam, Shekhar; Ranvir, Ramchandra; Patel, Harilal; Sundar, Rajesh; Jain, Mukul

Femtosecond laser versus mechanical microkeratome use for laser‐assisted in‐situ keratomileusis (LASIK)

飞秒激光与机械微型角膜刀在激光辅助原位角膜磨镶术(LASIK)中的应用比较

Kansagra, Kevinkumar A; Parmar, Deven; Jani, Rajendra H; Srinivas, Nuggehally R; Lickliter, Jason; Patel, Harilal V; Parikh, Devang P; Heading, Heather; Patel, Hardik B; Gupta, Rahul J; Shah, Chintan Y; Patel, Maulik R; Dholakia, Vyom N; Sukhadiya, Raghav; Jain, Mukul R; Parmar, Krupi V; Barot, Kinjal; Kahuam‐López, Nicolás; Navas, Alejandro; Castillo‐Salgado, Carlos; Graue‐Hernandez, Enrique O; Jimenez‐Corona, Aida; Ibarra, Antonio

ZY15557, a novel, long acting inhibitor of dipeptidyl peptidase-4, for the treatment of Type 2 diabetes mellitus

ZY15557 是一种新型的长效二肽基肽酶-4抑制剂,用于治疗2型糖尿病。

Jain, Mukul R; Joharapurkar, Amit A; Kshirsagar, Samadhan G; Patel, Vishal J; Bahekar, Rajesh H; Patel, Harilal V; Jadav, Pradip A; Patel, Pankaj R; Desai, Ranjit C

Discovery of a Potent and Orally Efficacious TGR5 Receptor Agonist

发现一种强效且口服有效的TGR5受体激动剂

Agarwal, Sameer; Patil, Amit; Aware, Umesh; Deshmukh, Prashant; Darji, Brijesh; Sasane, Santosh; Sairam, Kalapatapu V V M; Priyadarsiny, Priyanka; Giri, Poonam; Patel, Harilal; Giri, Suresh; Jain, Mukul; Desai, Ranjit C