日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of a Covalent Importin-5 Inhibitor, Goyazensolide, from a Collective Synthesis of Furanoheliangolides

通过呋喃杂环己烷内酯的集体合成鉴定出共价型 Importin-5 抑制剂 Goyazensolide

Liu, Weilong; Patouret, Rémi; Barluenga, Sofia; Plank, Michael; Loewith, Robbie; Winssinger, Nicolas

Correction: HDX-MS reveals structural determinants for RORγ hyperactivation by synthetic agonists

更正:HDX-MS揭示了合成激动剂过度激活RORγ的结构决定因素

Strutzenberg, Timothy S; Garcia-Ordonez, Ruben D; Novick, Scott J; Park, HaJeung; Chang, Mi Ra; Doebellin, Christelle; He, Yuanjun; Patouret, Rémi; Kamenecka, Theodore M; Griffin, Patrick R

HDX-MS reveals structural determinants for RORγ hyperactivation by synthetic agonists

HDX-MS 揭示了合成激动剂导致 RORγ 过度活化的结构决定因素

Timothy S Strutzenberg, Ruben D Garcia-Ordonez, Scott J Novick, HaJeung Park, Mi Ra Chang, Christelle Doebellin, Yuanjun He, Rémi Patouret, Theodore M Kamenecka, Patrick R Griffin

Identification of an aminothiazole series of RORβ modulators

鉴定一类氨基噻唑类RORβ调节剂

Patouret, Rémi; Doebelin, Christelle; Garcia-Ordonez, Ruben D; Chang, Mi Ra; Ruiz, Claudia; Cameron, Michael D; Griffin, Patrick R; Kamenecka, Theodore M

Design, synthesis, and evaluation of simple phenol amides as ERRγ agonists

设计、合成和评价简单的酚酰胺类化合物作为ERRγ激动剂

Lin, Hua; Doebelin, Christelle; Patouret, Rémi; Garcia-Ordonez, Ruben D; Chang, M R; Dharmarajan, Venkatasubramanian; Bayona, Claudia Ruiz; Cameron, Michael D; Griffin, Patrick R; Kamenecka, Theodore M

Identification of potent RORβ modulators: Scaffold variation

鉴定有效的RORβ调节剂:支架变异

Doebelin, Christelle; Patouret, Rémi; Garcia-Ordonez, Ruben D; Chang, Mi Ra; Dharmarajan, Venkatasubramanian; Novick, Scott; Ciesla, Anthony; Campbell, Sean; Solt, Laura A; Griffin, Patrick R; Kamenecka, Theodore M

N-Arylsulfonyl Indolines as Retinoic Acid Receptor-Related Orphan Receptor γ (RORγ) Agonists

N-芳基磺酰基吲哚啉类化合物作为视黄酸受体相关孤儿受体γ (RORγ) 激动剂

Doebelin, Christelle; Patouret, Rémi; Garcia-Ordonez, Ruben D; Chang, Mi Ra; Dharmarajan, Venkatasubramanian; Kuruvilla, Dana S; Novick, Scott J; Lin, Li; Cameron, Michael D; Griffin, Patrick R; Kamenecka, Theodore M

Synthesis of 2-aryl-2H-tetrazoles via a regioselective [3+2] cycloaddition reaction

通过区域选择性[3+2]环加成反应合成2-芳基-2H-四唑

Patouret, Remi; Kamenecka, Theodore M